SCHEMBL5609138

SCHEMBL5609138

COc1c(-c2ccccc2)cccc1C1OCCO1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.36
PDE4A P27815 2/20 0.36
PDE4C Q08493 2/20 0.36
PDE4D Q08499 2/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
USP30 Q70CQ3 1/20 0.35
FABP3 P05413 1/20 0.35
NR1H4 Q96RI1 1/20 0.35
CYP19A1 P11511 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
NR3C1 P04150 1/20 0.35
HTR1A P08908 1/20 0.35
HTR7 P34969 1/20 0.35
HTR2B P41595 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1256101 0.81 ADRA2A (0.41) CHRNB2CHRNA4USP30ADRA1DADRA1A
SCHEMBL18085976 0.78 NPC1 (0.37) NPC1RAB9AHTR2BADRA1A
SCHEMBL13385087 0.76 PDE4B (0.48) PDE4BPDE4APDE4CPDE4DNR1H4
SCHEMBL18288005 0.74 RAB9A (0.40) NPC1RAB9AKDM4EADRA1A
SCHEMBL18555663 0.72 KDM4E (0.41) CYP19A1KDM4ELMNAADRA1DADRA1A
SCHEMBL6231988 0.72 SMN1; SMN2 (0.39) NPC1RAB9AKDM4ELMNA
SCHEMBL10761583 0.72 HTR2C (0.49) CYP19A1HTR2B
SCHEMBL28039230 0.70 PDE4B (0.50) PDE4BPDE4APDE4CPDE4DKDM4E
SCHEMBL28923075 0.70 CYP1A1 (0.42) NPC1RAB9AKDM4E
SCHEMBL3727526 0.70 TSHR (0.36) NPC1RAB9AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1354887-B1 Ligands for metals and improved metal-catalyzed processes based thereon MASSACHUSETTS INST TECHNOLOGY (US) 2007-04-25 EP disclosed
EP-1097158-B1 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INST TECHNOLOGY (US) 2006-01-25 EP disclosed
EP-1354887-A1 Ligands for metals and improved metal-catalyzed processes based thereon Massachusetts Insitute of Technology (US) 2003-10-22 EP disclosed
EP-1097158-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2001-05-09 EP disclosed
WO-2000002887-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2000-01-20 WO disclosed