SCHEMBL10769983

SCHEMBL10769983

OC1=Cc2ccccc2SC=C1

nearest known ligand 0.31

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7520710 0.73 DAO (0.31) GPR84
SCHEMBL7922049 0.72 TSHR (0.33)
SCHEMBL348197 0.67
Water SCHEMBL19745732 0.65
Water SCHEMBL19744946 0.65
SCHEMBL563542 0.65 KDM4E (0.35) GPR84
SCHEMBL493616 0.64 TRPA1 (0.30)
SCHEMBL4832141 0.62 MEN1 (0.41) GPR84
SCHEMBL4832146 0.62 MEN1 (0.41) GPR84
SCHEMBL2937188 0.62 ACHE (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112204035-A Substituted 3,4,12,12 a-tetrahydro-1 n1- [1,4] oxazino [3,4-c ] pyrido [2,1-f ] [1,2,4] triazine-6, 8-diones, pharmaceutical compositions, methods of production and uses thereof 亚历山大·瓦西里耶维奇·伊瓦切恩科 2021-01-08 CN claimed
WO-2020226532-A1 SUBSTITUTED 3,4,12,12A-TETRAHYDRO-1H-[1,4]OXAZINO[3,4-C]PYRIDO[2,1-F][1,2,4]TRIAZINE-6,8-DIONE, PHARMACEUTICAL COMPOSITION, AND METHODS FOR PREPARING AND USING SAME ИВАЩЕНКО, Александр Васильевич 2020-11-12 WO claimed
CN-112204035-A Substituted 3,4,12,12 a-tetrahydro-1 n1- [1,4] oxazino [3,4-c ] pyrido [2,1-f ] [1,2,4] triazine-6, 8-diones, pharmaceutical compositions, methods of production and uses thereof 亚历山大·瓦西里耶维奇·伊瓦切恩科 2021-01-08 CN disclosed
WO-2020226532-A1 SUBSTITUTED 3,4,12,12A-TETRAHYDRO-1H-[1,4]OXAZINO[3,4-C]PYRIDO[2,1-F][1,2,4]TRIAZINE-6,8-DIONE, PHARMACEUTICAL COMPOSITION, AND METHODS FOR PREPARING AND USING SAME ИВАЩЕНКО, Александр Васильевич 2020-11-12 WO disclosed
EP-0226320-A1 Imidazolyl thieno-benzothiepin derivatives and processes for the preparation thereof SPOFA Spojené Podniky Pro Zdravotnickou Vyrobu (CS) 1987-06-24 EP disclosed