SCHEMBL10770909

SCHEMBL10770909

COC(=O)c1ccc(C(CCC(=O)N(C)C)c2c[nH]c3ccc(C(=O)NCC4CCCC4)cc23)c(OC)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.42
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HTR4 Q13639 2/20 0.38
ROCK2 O75116 3/20 0.38
ROCK1 Q13464 2/20 0.38
PDE4A P27815 2/20 0.37
PDE4B Q07343 2/20 0.37
PDE4C Q08493 2/20 0.37
PDE4D Q08499 2/20 0.37
HTT P42858 1/20 0.37
ATM Q13315 1/20 0.36
TRPV1 Q8NER1 2/20 0.36
KDM4E B2RXH2 1/20 0.36
THRB P10828 1/20 0.36
HPGD P15428 1/20 0.36
MAPK14 Q16539 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9667839 0.91 TDP1 (0.43) TDP1ALDH1A1LMNASMN1; SMN2HTR4
SCHEMBL9669473 0.85 TDP1 (0.43) TDP1ALDH1A1LMNASMN1; SMN2HTR4
SCHEMBL9669804 0.85 TDP1 (0.48) TDP1ALDH1A1LMNASMN1; SMN2HTR4
SCHEMBL8998195 0.84 TDP1 (0.42) TDP1ALDH1A1LMNASMN1; SMN2HTR4
SCHEMBL9669675 0.80 ALDH1A1 (0.42) TDP1ALDH1A1LMNASMN1; SMN2HTR4
SCHEMBL9669740 0.80 TDP1 (0.48) TDP1ALDH1A1LMNASMN1; SMN2HTR4
SCHEMBL8998143 0.79 TDP1 (0.42) TDP1ALDH1A1LMNASMN1; SMN2HTR4
SCHEMBL9668025 0.78 CYSLTR2 (0.43) ALDH1A1LMNASMN1; SMN2
SCHEMBL8951236 0.77 CYSLTR2 (0.44) ALDH1A1LMNAKDM4E
SCHEMBL8998166 0.76 GPR84 (0.55) TDP1HTR4ROCK2ROCK1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0227241-A2 Medicinal indole and indazole keto sulphone derivatives ZENECA INC. (US) 1987-07-01 EP disclosed