SCHEMBL1079351

SCHEMBL1079351

CCCC(C)C(C(=O)Nc1cccc(CC(C(=O)O)C(C)(C)C)c1C)c1ccc(CN2N=C(c3ccccc3)OCC2=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGES O14684 7/20 0.38
PTGS2 P35354 12/20 0.34
MRGPRX1 Q96LB2 1/20 0.32
MAOB P27338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3694861 0.93 PTGS2 (0.37) PTGESPTGS2MRGPRX1MAOB
SCHEMBL3697908 0.91 PTGES (0.36) PTGESPTGS2MRGPRX1
SCHEMBL3704804 0.91 PTGES (0.36) PTGESPTGS2MRGPRX1MAOB
SCHEMBL3694433 0.90 PTGS2 (0.36) PTGESPTGS2MRGPRX1
SCHEMBL1081379 0.88 PTGES (0.51) PTGESPTGS2
SCHEMBL1079353 0.86 PTGES (0.43) PTGESPTGS2
SCHEMBL1081836 0.86 PTGES (0.45) PTGESPTGS2MRGPRX1MAOB
SCHEMBL1080114 0.85 SMN1; SMN2 (0.37) PTGES
SCHEMBL1177252 0.85 PTGS2 (0.50) PTGESPTGS2
SCHEMBL3700948 0.83 MAOB (0.34) PTGESMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268625-B1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF Bayer Pharma AG (DE) 2012-05-16 EP disclosed
EP-2268625-A1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF Bayer Schering Pharma Aktiengesellschaft (DE) 2011-01-05 EP disclosed
WO-2009127338-A1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-10-22 WO disclosed