SCHEMBL3697908

SCHEMBL3697908

COCC(C)C(C(=O)Nc1cccc(CC(C(=O)O)C(C)(C)C)c1C)c1ccc(CN2N=C(c3ccccc3)OCC2=O)cc1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGES O14684 4/20 0.36
PTGS2 P35354 11/20 0.34
PDCD1 Q15116 4/20 0.34
CD274 Q9NZQ7 4/20 0.34
MRGPRX1 Q96LB2 1/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3694861 0.93 PTGS2 (0.37) PTGESPTGS2MRGPRX1PPARGPPARA
SCHEMBL1079351 0.91 PTGES (0.38) PTGESPTGS2MRGPRX1
SCHEMBL3704804 0.90 PTGES (0.36) PTGESPTGS2MRGPRX1
SCHEMBL3694433 0.89 PTGS2 (0.36) PTGESPTGS2MRGPRX1
SCHEMBL1078521 0.88 PTGES (0.49) PTGESPTGS2
SCHEMBL1178914 0.87 PTGES (0.41) PTGESPTGS2
SCHEMBL1177252 0.84 PTGS2 (0.50) PTGESPTGS2
SCHEMBL1081836 0.84 PTGES (0.45) PTGESPTGS2MRGPRX1PPARG
SCHEMBL3700948 0.83 MAOB (0.34) PTGES
SCHEMBL1069734 0.81 PTGS2 (0.33) PTGESPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268625-B1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF Bayer Pharma AG (DE) 2012-05-16 EP disclosed