SCHEMBL3704804

SCHEMBL3704804

Cc1c(CC(C(=O)O)C(C)(C)C)cccc1NC(=O)C(c1ccc(CN2N=C(c3ccccc3)OCC2=O)cc1)C(C)CC#N

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGES O14684 3/20 0.36
PTGS2 P35354 9/20 0.35
MAOB P27338 1/20 0.34
KMT2A Q03164 1/20 0.33
MRGPRX1 Q96LB2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3694861 0.92 PTGS2 (0.37) PTGESPTGS2MAOBMRGPRX1
SCHEMBL1079351 0.91 PTGES (0.38) PTGESPTGS2MAOBMRGPRX1
SCHEMBL3697908 0.90 PTGES (0.36) PTGESPTGS2MRGPRX1
SCHEMBL3694433 0.89 PTGS2 (0.36) PTGESPTGS2MRGPRX1
SCHEMBL1177996 0.88 PTGES (0.48) PTGESPTGS2
SCHEMBL1178612 0.87 PTGES (0.40) PTGESPTGS2MAOB
SCHEMBL1177252 0.83 PTGS2 (0.50) PTGESPTGS2
SCHEMBL1081836 0.83 PTGES (0.45) PTGESPTGS2MAOBMRGPRX1
SCHEMBL3700948 0.82 MAOB (0.34) PTGESMAOB
SCHEMBL3695678 0.81 KMT2A (0.43) MAOBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268625-B1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF Bayer Pharma AG (DE) 2012-05-16 EP disclosed