SCHEMBL10795296

SCHEMBL10795296

CCSC1=NO[C@H](CNC(=O)[C@H](CC(=O)O)N(Cc2ccccc2)C(=O)OCc2ccccc2)C1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 7/20 0.44
CYP1A2 P05177 1/20 0.37
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
EPOR P19235 2/20 0.35
ITGB3 P05106 8/20 0.34
ITGA2B P08514 5/20 0.34
MME P08473 1/20 0.34
ACE P12821 1/20 0.34
ECE1 P42892 1/20 0.34
ITGAV P06756 7/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9825943 0.82 TGM2 (0.59) TGM2CYP1A2ITGB3ITGAV
SCHEMBL9825615 0.81 TGM2 (0.44) TGM2CYP1A2ALDH1A1ITGB3ITGA2B
SCHEMBL9826404 0.78 TGM2 (0.44) TGM2CYP1A2ITGB3ITGA2BMME
SCHEMBL9825336 0.78 TGM2 (0.69) TGM2CYP1A2
SCHEMBL9826397 0.78 TGM2 (0.69) TGM2CYP1A2
SCHEMBL9825407 0.78 TGM2 (0.42) TGM2CYP1A2ALDH1A1HSD17B10ITGB3
SCHEMBL9825638 0.77 TGM2 (0.57) TGM2CYP1A2ITGB3ITGA2BITGAV
SCHEMBL9826129 0.77 CTSL (0.54) TGM2CYP1A2LMNAITGB3ITGAV
SCHEMBL9825517 0.77 TGM2 (0.75) TGM2
SCHEMBL9825735 0.76 CTSL (0.56) TGM2CYP1A2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0237082-A2 3,5-disubstituted 4,5-dihydroisoxazoles as transglutaminase inhibitors SYNTEX (U.S.A.) INC. (US) 1987-09-16 EP disclosed