SCHEMBL10797246

SCHEMBL10797246

O=S(=O)(c1ccccc1)C1CCCNCC1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.46
KCNH2 Q12809 2/20 0.44
HTR2C P28335 1/20 0.44
MAPT P10636 2/20 0.42
HTR6 P50406 7/20 0.42
MMP8 P22894 2/20 0.41
MMP13 P45452 2/20 0.41
MMP1 P03956 1/20 0.41
GBA1 P04062 1/20 0.41
SLC18A3 Q16572 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17803 0.93 HTR2A (0.51) HTR2AKCNH2HTR2CMAPTHTR6
Hydrochloric Acid SCHEMBL1021139 0.91 HTR2A (0.50) HTR2AKCNH2HTR2CMAPTHTR6
SCHEMBL711807 0.86 APLNR (0.50) HTR2AKCNH2HTR2CMAPTHTR6
Hydrochloric Acid SCHEMBL28532829 0.85 APLNR (0.49) HTR2AKCNH2HTR2CMAPTHTR6
SCHEMBL14501834 0.83 HTR6 (0.40) HTR6MMP8MMP13MMP1ALDH1A1
SCHEMBL777971 0.83 MAPT (0.56) HTR2AKCNH2HTR2CMAPTHTR6
SCHEMBL7541817 0.83 HTR2A (0.56) HTR2AKCNH2HTR2CMAPTHTR6
SCHEMBL336837 0.82 HTR2A (0.45) HTR2AKCNH2HTR2CMAPTHTR6
SCHEMBL10799767 0.81 MAPT (0.45) HTR2AKCNH2HTR2CMAPTHTR6
SCHEMBL776895 0.81 MAPT (0.55) HTR2AKCNH2HTR2CMAPTHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4642348-A ANTIARRHYTHMIA AGENTS A. H. ROBINS COMPANY, INCORPORATED (US) 1987-02-10 US disclosed
US-4593102-A N-[(amino)alkyl]-1-pyrrolidine, 1-piperidine and 1-homopiperidinecarboxamides (and thiocarboxamides) with sulfur linked substitution in the 2, 3 or 4-position A. H. ROBINS COMPANY, INC. (US) 1986-06-03 US disclosed
EP-0160436-A2 N-[(Amino)Alkyl]-1-pyrrolidine, 1-piperidine and 1-homopiperidinecarboxamides (and thiocarboxamides) with sulphur linked substitution in the 2, 3 or 4-position A.H. ROBINS COMPANY, INCORPORATED (US) 1985-11-06 EP disclosed