SCHEMBL10798157

SCHEMBL10798157

O=S(=O)(c1cccc2c1CCC2)C1CCCNC1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
APLNR P35414 2/20 0.41
METAP2 P50579 2/20 0.38
CXCR2 P25025 10/20 0.38
CX3CR1 P49238 1/20 0.35
HTR6 P50406 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10797930 0.99 APLNR (0.40) APLNRMETAP2CXCR2CX3CR1HTR6
SCHEMBL10795662 0.78 METAP2 (0.45) METAP2HTR6
SCHEMBL10798931 0.78 APLNR (0.38) APLNRMETAP2CXCR2
SCHEMBL10795182 0.78 CXCR2 (0.43) APLNRCXCR2CX3CR1HTR6
Hydrochloric Acid SCHEMBL10797733 0.77 METAP2 (0.44) METAP2
Hydrochloric Acid SCHEMBL10800177 0.77 CXCR2 (0.42) APLNRCXCR2CX3CR1HTR6
SCHEMBL10794598 0.75 HTR6 (0.54) APLNRHTR6
Hydrochloric Acid SCHEMBL10795401 0.74 HTR6 (0.53) APLNRHTR6
SCHEMBL10795334 0.74 DRD2 (0.42) APLNRCXCR2HTR6
SCHEMBL10795383 0.72 CA12 (0.47) APLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4642348-A ANTIARRHYTHMIA AGENTS A. H. ROBINS COMPANY, INCORPORATED (US) 1987-02-10 US disclosed
US-4593102-A N-[(amino)alkyl]-1-pyrrolidine, 1-piperidine and 1-homopiperidinecarboxamides (and thiocarboxamides) with sulfur linked substitution in the 2, 3 or 4-position A. H. ROBINS COMPANY, INC. (US) 1986-06-03 US disclosed
EP-0160436-A2 N-[(Amino)Alkyl]-1-pyrrolidine, 1-piperidine and 1-homopiperidinecarboxamides (and thiocarboxamides) with sulphur linked substitution in the 2, 3 or 4-position A.H. ROBINS COMPANY, INCORPORATED (US) 1985-11-06 EP disclosed