SCHEMBL10799648

SCHEMBL10799648

O=C(O)C1CN(CC2CCCCC2)CCC1=O

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.42
ADRA2C P18825 1/20 0.42
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
F2R P25116 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CCR1 P32246 2/20 0.40
ACHE P22303 1/20 0.38
SIGMAR1 Q99720 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPK1 P28482 1/20 0.37
GRM2 Q14416 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
OPRL1 P41146 1/20 0.37
KDM2B Q8NHM5 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6583721 0.81 ALDH1A1 (0.40) CHRM5SMN1; SMN2
Hydrochloric Acid SCHEMBL10945868 0.80 ALDH1A1 (0.40) CHRM5SMN1; SMN2
SCHEMBL23002177 0.76 ITGB3 (0.35) CHRM5ITGB3ITGA2BF2RSMN1; SMN2
Hydrochloric Acid SCHEMBL442313 0.74 CYP3A4 (0.35) CHRM5ITGB3ITGA2BF2RSMN1; SMN2
SCHEMBL7425201 0.73 SMN1; SMN2 (0.39) SMN1; SMN2KDM2B
SCHEMBL29896656 0.72 MAPT (0.42) CHRM5SMN1; SMN2KDM4EKDM2B
SCHEMBL27584327 0.71 CHRM5 (0.52) CHRM5ADRA2CSMN1; SMN2KDM4EMAPK1
SCHEMBL16102614 0.71 CHRM5 (0.61) CHRM5ADRA2CSMN1; SMN2ACHESIGMAR1
SCHEMBL6583551 0.71 CHRM5 (0.61) CHRM5ADRA2CSMN1; SMN2ACHESIGMAR1
SCHEMBL3009112 0.71 CHRM5 (0.61) CHRM5ADRA2CSMN1; SMN2ACHESIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0099303-B1 BENZOTHIOPYRANOPYRIDINONES AND THEIR SALTS, THEIR PREPARATION AND USE AS MEDICAMENTS, AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1987-08-19 EP disclosed
EP-0099303-A2 Benzothiopyranopyridinones and their salts, their preparation and use as medicaments, and compositions containing them ROUSSEL-UCLAF (FR) 1984-01-25 EP disclosed