SCHEMBL10815249

SCHEMBL10815249

NC1CC2CCCC(C1)N2Cc1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CXCR6 O00574 1/20 0.46
OPRK1 P41145 2/20 0.43
DRD2 P14416 2/20 0.43
DRD4 P21917 2/20 0.43
DRD3 P35462 1/20 0.43
ARG1 P05089 1/20 0.42
ARG2 P78540 1/20 0.42
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LTA4H P09960 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3881487 0.93 DRD2 (0.48) CXCR6DRD2DRD4DRD3ARG1
SCHEMBL3881484 0.93 DRD2 (0.48) CXCR6DRD2DRD4DRD3ARG1
SCHEMBL30833195 0.93 DRD2 (0.48) CXCR6DRD2DRD4DRD3ARG1
SCHEMBL10817485 0.85 OPRK1 (0.52) OPRK1DRD2DRD4DRD3MAPT
SCHEMBL10812514 0.85 OPRK1 (0.58) OPRK1MAPTALDH1A1
SCHEMBL9023345 0.85 CHRM2 (0.54) OPRK1ALDH1A1LMNA
SCHEMBL8120312 0.85 CHRM2 (0.54) OPRK1ALDH1A1LMNA
SCHEMBL20967986 0.85 CHRM2 (0.54) OPRK1ALDH1A1LMNA
SCHEMBL27676903 0.84 DRD2 (0.51) CXCR6OPRK1DRD2DRD4DRD3
SCHEMBL9413102 0.82 DRD4 (0.47) CXCR6DRD2DRD4DRD3ARG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0076592-B1 AZABICYCLO-(3,3,1)-NONYLBENZAMIDE DERIVATIVES, PROCESSES FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1987-01-28 EP disclosed
US-4560757-A 9-Azabicyclo(3.3.1) nonane intermediates for compounds useful in the treatment of CNS disorders BEECHAM GROUP P.L.C. (GB) 1985-12-24 US disclosed
US-4472413-A PSYCHOLOGICAL DISORDERS BEECHAM GROUP P.L.C. (GB) 1984-09-18 US disclosed