SCHEMBL10832467

SCHEMBL10832467

CCc1nc(-c2ccc(Cl)cc2)c(C)o1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TARBP2 Q15633 1/20 0.41
RXRA P19793 3/20 0.40
RXRB P28702 3/20 0.40
RXRG P48443 3/20 0.40
HTT P42858 1/20 0.39
KMT2A Q03164 3/20 0.38
ALOX12 P18054 1/20 0.38
CRHR1 P34998 1/20 0.38
ALDH1A1 P00352 4/20 0.37
LMNA P02545 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 2/20 0.37
SLC22A1 O15245 1/20 0.37
DHFR P00374 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
HEXA P06865 1/20 0.37
HEXB P07686 1/20 0.37
CYP3A4 P08684 1/20 0.37
HTR1A P08908 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15578164 0.83 NPC1 (0.40) KMT2AALDH1A1KDM4EMEN1TP53
SCHEMBL10269662 0.82 KDM4E (0.50) RXRARXRBRXRGALDH1A1LMNA
SCHEMBL9848741 0.80 SIRT2 (0.54) TARBP2RXRARXRBRXRGKMT2A
SCHEMBL9440740 0.79 SIRT2 (0.47) TARBP2RXRARXRBRXRGHTT
SCHEMBL10833341 0.79 RXRA (0.37) RXRARXRBRXRGHTTKMT2A
SCHEMBL9441135 0.78 RAB9A (0.52) TARBP2HTTKMT2AALDH1A1LMNA
SCHEMBL5536993 0.78 ALDH1A1 (0.47) TARBP2ALDH1A1LMNAKDM4EHTR2A
SCHEMBL3914104 0.76 ALDH1A1 (0.43) TARBP2HTTKMT2AALOX12CRHR1
SCHEMBL10834263 0.72 MAOA (0.44) RXRARXRBRXRGKMT2AALDH1A1
SCHEMBL10834256 0.72 RXRA (0.58) RXRARXRBRXRGHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4596816-A Pharmaceuticals TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1986-06-24 US disclosed
EP-0092239-A2 Oxazole derivatives, production and use thereof Takeda Chemical Industries, Ltd. (JP) 1983-10-26 EP disclosed