SCHEMBL1083353

SCHEMBL1083353

C=Cc1cc2ccc(OC)cc2nc1OC1CN(C(=O)OC(C)(C)C)C(C)(C(=O)O)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.36
KDM4E B2RXH2 3/20 0.36
NPC1 O15118 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
HPGDS O60760 6/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
BACE1 P56817 1/20 0.34
PIK3CD O00329 2/20 0.33
PIK3CA P42336 2/20 0.33
PIK3CB P42338 2/20 0.33
PIK3CG P48736 2/20 0.33
DYRK1A Q13627 1/20 0.32
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
SLC2A1 P11166 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1072471 1.00 RAB9A (0.36) RAB9AKDM4ENPC1L3MBTL1HPGDS
SCHEMBL1072580 0.89 RAB9A (0.36) RAB9AKDM4ENPC1L3MBTL1HPGDS
SCHEMBL21800693 0.84 BACE1 (0.34) RAB9AKDM4ENPC1L3MBTL1HPGDS
SCHEMBL3305756 0.84 SLC2A1 (0.33) RAB9AKDM4ENPC1L3MBTL1BACE1
SCHEMBL1583415 0.84 BACE1 (0.37) RAB9AKDM4ENPC1L3MBTL1HPGDS
SCHEMBL21800783 0.83 BACE1 (0.34) RAB9AKDM4ENPC1L3MBTL1HPGDS
SCHEMBL12934504 0.78 RAB9A (0.44) RAB9AKDM4ENPC1L3MBTL1PPARD
SCHEMBL2427449 0.77 PIK3CD (0.38) PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL3302407 0.77 GPR119 (0.36) KDM4E
SCHEMBL1068681 0.77 KDM4E (0.36) RAB9AKDM4ENPC1L3MBTL1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268285-A1 THERAPEUTIC COMPOUNDS Merck Sharp & Dohme Corp. (US) 2011-01-05 EP disclosed