SCHEMBL10835355

SCHEMBL10835355

COc1ccc(F)cc1N1CCN(CCCN2C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.79
DRD3 P35462 6/20 0.79
HTR1A P08908 7/20 0.76
ALDH1A1 P00352 2/20 0.76
HTR7 P34969 2/20 0.76
MEN1 O00255 1/20 0.76
CYP3A4 P08684 1/20 0.76
CYP2D6 P10635 1/20 0.76
ALOX12 P18054 1/20 0.76
ADRA1D P25100 1/20 0.76
ADRA1A P35348 1/20 0.76
ADRA1B P35368 1/20 0.76
KMT2A Q03164 1/20 0.76
HIF1A Q16665 1/20 0.76
HSD17B10 Q99714 1/20 0.76
KDM4E B2RXH2 1/20 0.74
GLA P06280 1/20 0.74
HPGD P15428 1/20 0.74
HTR2A P28223 1/20 0.63
HTR6 P50406 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10835477 0.91 DRD2 (0.79) DRD2DRD3HTR1AALDH1A1HTR7
SCHEMBL10835973 0.89 DRD2 (1.00) DRD2DRD3HTR1AALDH1A1HTR7
SCHEMBL6771089 0.87 DRD2 (0.76) DRD2DRD3HTR1AALDH1A1HTR7
Nan-190 SCHEMBL30080779 0.86 HTR1A (1.00) DRD2DRD3HTR1AALDH1A1HTR7
Nan-190 SCHEMBL2231820 0.86 HTR1A (1.00) DRD2DRD3HTR1AALDH1A1HTR7
Nan-190 SCHEMBL29389115 0.86 HTR1A (1.00) DRD2DRD3HTR1AALDH1A1HTR7
Nan-190 SCHEMBL29390376 0.85 ALDH1A1 (1.00) DRD2DRD3HTR1AALDH1A1HTR7
SCHEMBL14761599 0.85 HTR1A (0.98) DRD2DRD3HTR1AALDH1A1HTR7
Nan-190 SCHEMBL4083153 0.85 ALDH1A1 (1.00) DRD2DRD3HTR1AALDH1A1HTR7
SCHEMBL5423795 0.85 DRD2 (0.57) DRD2DRD3HTR1AALDH1A1HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4585773-A DIURETIC, HYPOTENSIVE BRISTOL-MYERS COMPANY (US) 1986-04-29 US disclosed