SCHEMBL10836282

SCHEMBL10836282

O=C1CCc2cc(C(O)CCN3CCN(c4ccccc4)CC3)ccc2N1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.56
ATM Q13315 1/20 0.56
GRIN2B Q13224 1/20 0.54
DRD2 P14416 2/20 0.53
HTR1A P08908 9/20 0.51
HTR2A P28223 2/20 0.51
KCNH2 Q12809 3/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
TP53 P04637 1/20 0.46
ALOX15 P16050 1/20 0.46
OGT O15294 1/20 0.45
HTR7 P34969 2/20 0.45
DRD4 P21917 1/20 0.45
DRD3 P35462 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10837291 0.95 DRD2 (0.57) ALDH1A1ATMGRIN2BDRD2HTR1A
SCHEMBL10835956 0.90 KCNH2 (0.50) ALDH1A1ATMGRIN2BDRD2HTR1A
SCHEMBL10837913 0.85 DRD2 (0.53) DRD2HTR1AHTR2AKCNH2DRD4
SCHEMBL10836115 0.85 KCNH2 (0.66) GRIN2BDRD2HTR1AHTR2AKCNH2
SCHEMBL10835827 0.85 DRD2 (0.51) ALDH1A1ATMGRIN2BDRD2HTR1A
SCHEMBL10835876 0.85 GRIN2B (0.54) GRIN2BDRD2HTR1AHTR2AKCNH2
SCHEMBL8549343 0.84 GRIN2B (0.59) GRIN2BMEN1KMT2AOGT
SCHEMBL10837721 0.83 HTR1A (0.65) DRD2HTR1AALOX15DRD4DRD3
SCHEMBL10837209 0.82 DRD2 (0.57) ALDH1A1GRIN2BDRD2HTR1AHTR2A
SCHEMBL10838656 0.82 GRIN2B (0.51) GRIN2BDRD2HTR1AHTR2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4619932-A CENTRAL NERVOUS SYSTEM CONTROLLERS; ANTI-SCHIZOPHRENIA AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1986-10-28 US disclosed
US-4605431-A ANTIDOTES FOR THIOLCARBAMATE HERBICIDES; PLANT SAFENING AGENTS MONSANTO COMPANY (US) 1986-08-12 US disclosed
US-4567187-A CENTRAL NERVOUS SYSTEM OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1986-01-28 US disclosed
US-4460593-A Carbostyril derivatives, and central nervous system controlling agents containing the carbostyril derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-07-17 US disclosed
US-4455422-A ANTIHISTAMINES, CNS CONTROLLERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-19 US disclosed