SCHEMBL10853166

SCHEMBL10853166

N=C(N)N(C(=O)NC1CCCCC1)c1cccnc1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.53
ALDH1A1 P00352 7/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
PKM P14618 1/20 0.47
TSHR P16473 3/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
EPHX1 P07099 1/20 0.42
USP2 O75604 1/20 0.41
LMNA P02545 2/20 0.40
HTT P42858 1/20 0.40
WNT1 P04628 1/20 0.39
DYRK1A Q13627 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10854108 0.96 POLB (0.48) POLBALDH1A1SMN1; SMN2PKMTSHR
SCHEMBL10857082 0.78 ALDH1A1 (0.41) ALDH1A1CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL10857092 0.77 PTGES (0.40) POLBALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL10855623 0.74 RECQL (0.41) POLBALDH1A1PKMHTT
SCHEMBL10857588 0.74 SYK (0.43) ALDH1A1CYP3A4CYP2C9LMNADYRK1A
SCHEMBL10852959 0.72 ALDH1A1 (0.50) POLBALDH1A1SMN1; SMN2PKMTSHR
Hydrochloric Acid SCHEMBL11555928 0.72 EPHX1 (0.49) SMN1; SMN2PKMCYP2C19EPHX1LMNA
SCHEMBL10857088 0.72 RECQL (0.40) ALDH1A1CYP3A4CYP2C9HTT
Hydrochloric Acid SCHEMBL11558867 0.72 EPHX1 (0.49) SMN1; SMN2PKMCYP2C19EPHX1LMNA
SCHEMBL27564720 0.72 POLB (0.45) POLBALDH1A1SMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4565826-A HYPOTENSIVE, CARDIONASCULAR, ANTIULCER, ANTISECRETORY, GASTROINTESTINAL DISORDERS WILLIAM H. RORER, INC. (US) 1986-01-21 US disclosed
US-4436911-A HYPOTENSIVE, ANTISPASMODIC, ANTIULCER, ANTIPARASITIC WILLIAM H. RORER, INC. (US) 1984-03-13 US disclosed