SCHEMBL10857082

SCHEMBL10857082

CNC(=O)N(C(=N)N)c1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
F7 P08709 1/20 0.40
F3 P13726 1/20 0.40
SARM1 Q6SZW1 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
SIRT6 Q8N6T7 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
SIRT3 Q9NTG7 1/20 0.40
SIRT5 Q9NXA8 1/20 0.40
SIRT4 Q9Y6E7 1/20 0.40
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
MKNK1 Q9BUB5 3/20 0.39
MKNK2 Q9HBH9 3/20 0.39
RECQL P46063 1/20 0.38
HTT P42858 1/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10857092 0.85 PTGES (0.40) ALDH1A1F7F3SARM1SIRT2
SCHEMBL10855623 0.85 RECQL (0.41) ALDH1A1F7F3SARM1SIRT2
SCHEMBL10857588 0.85 SYK (0.43) ALDH1A1F7F3SARM1SIRT2
SCHEMBL10857088 0.82 RECQL (0.40) ALDH1A1GAAHPGDMKNK1MKNK2
SCHEMBL10857210 0.81 CA1 (0.37) ALDH1A1SIRT3GAAHPGDCYP1A2
SCHEMBL10854337 0.81 RECQL (0.39) ALDH1A1F7F3SARM1SIRT2
SCHEMBL10852319 0.81 RECQL (0.39) ALDH1A1F7F3SARM1SIRT2
SCHEMBL11238745 0.81 LMNA (0.38) ALDH1A1SIRT2L3MBTL1LMNA
SCHEMBL10856096 0.80 HDAC3 (0.44) ALDH1A1HPGDRECQLNPC1RAB9A
SCHEMBL10860776 0.79 MAPT (0.44) ALDH1A1GAAL3MBTL1THRBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4565826-A HYPOTENSIVE, CARDIONASCULAR, ANTIULCER, ANTISECRETORY, GASTROINTESTINAL DISORDERS WILLIAM H. RORER, INC. (US) 1986-01-21 US disclosed
US-4436911-A HYPOTENSIVE, ANTISPASMODIC, ANTIULCER, ANTIPARASITIC WILLIAM H. RORER, INC. (US) 1984-03-13 US disclosed