SCHEMBL10857092

SCHEMBL10857092

CC(C)NC(=O)N(C(=N)N)c1cccnc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 3/20 0.40
ALDH1A1 P00352 1/20 0.38
AKR1C3 P42330 2/20 0.38
F7 P08709 1/20 0.37
F3 P13726 1/20 0.37
SARM1 Q6SZW1 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.37
SIRT6 Q8N6T7 1/20 0.37
SIRT1 Q96EB6 1/20 0.37
SIRT3 Q9NTG7 1/20 0.37
SIRT5 Q9NXA8 1/20 0.37
SIRT4 Q9Y6E7 1/20 0.37
GAA P10253 2/20 0.37
HPGD P15428 1/20 0.37
POLB P06746 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP2C19 P33261 1/20 0.36
RECQL P46063 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10857082 0.85 ALDH1A1 (0.41) ALDH1A1F7F3SARM1SIRT2
SCHEMBL10852319 0.83 RECQL (0.39) ALDH1A1F7F3SARM1SIRT2
SCHEMBL10849103 0.83 MAOA (0.37) PTGESALDH1A1AKR1C3HPGDCYP3A4
SCHEMBL10855623 0.81 RECQL (0.41) ALDH1A1F7F3SARM1SIRT2
SCHEMBL10857588 0.81 SYK (0.43) ALDH1A1F7F3SARM1SIRT2
SCHEMBL10857088 0.79 RECQL (0.40) ALDH1A1GAAHPGDCYP3A4CYP2C9
SCHEMBL10854108 0.78 POLB (0.48) ALDH1A1POLBCYP3A4CYP2C9CYP2C19
SCHEMBL10854337 0.78 RECQL (0.39) ALDH1A1F7F3SARM1SIRT2
SCHEMBL10853166 0.77 POLB (0.53) ALDH1A1POLBCYP3A4CYP2C9CYP2C19
SCHEMBL10856096 0.77 HDAC3 (0.44) ALDH1A1HPGDPOLBCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4565826-A HYPOTENSIVE, CARDIONASCULAR, ANTIULCER, ANTISECRETORY, GASTROINTESTINAL DISORDERS WILLIAM H. RORER, INC. (US) 1986-01-21 US disclosed
US-4436911-A HYPOTENSIVE, ANTISPASMODIC, ANTIULCER, ANTIPARASITIC WILLIAM H. RORER, INC. (US) 1984-03-13 US disclosed