SCHEMBL10857049

SCHEMBL10857049

CNC(=N)NC(=O)Nc1ncco1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.46
FFAR2 O15552 1/20 0.40
CSNK2A2 P19784 1/20 0.36
CSNK2B P67870 1/20 0.36
CSNK2A1 P68400 1/20 0.36
CSNK2A3 Q8NEV1 1/20 0.36
NAMPT P43490 1/20 0.34
PSMD14 O00487 1/20 0.34
STAMBP O95630 1/20 0.34
COPS5 Q92905 1/20 0.34
LRRK2 Q5S007 1/20 0.32
IDH2 P48735 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26546183 0.83 EPHX2 (0.53) EPHX2FFAR2CSNK2A2CSNK2BCSNK2A1
SCHEMBL10854597 0.73 HTT (0.44) EPHX2FFAR2
SCHEMBL29128627 0.73 EPHX2 (0.47) EPHX2FFAR2CSNK2A2CSNK2BCSNK2A1
SCHEMBL17186398 0.72 EPHX2 (0.49) EPHX2FFAR2CSNK2A2CSNK2BCSNK2A1
SCHEMBL3262436 0.72
Hydrochloric Acid SCHEMBL17186463 0.71 EPHX2 (0.48) EPHX2FFAR2CSNK2A2CSNK2BCSNK2A1
SCHEMBL3070030 0.70
SCHEMBL10856446 0.70 KDM4C (0.43)
SCHEMBL10854078 0.70 NPC1 (0.30)
SCHEMBL10857203 0.69 MDM2 (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4565826-A HYPOTENSIVE, CARDIONASCULAR, ANTIULCER, ANTISECRETORY, GASTROINTESTINAL DISORDERS WILLIAM H. RORER, INC. (US) 1986-01-21 US disclosed
US-4436911-A HYPOTENSIVE, ANTISPASMODIC, ANTIULCER, ANTIPARASITIC WILLIAM H. RORER, INC. (US) 1984-03-13 US disclosed