SCHEMBL10875813

SCHEMBL10875813

O=C1C[C@H]2C(c3ccccc3)Cc3ccccc3[C@H]2CN1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP3 Q9Y6F1 1/20 0.43
SLC6A3 Q01959 3/20 0.40
MTNR1A P48039 1/20 0.39
MEN1 O00255 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
KMT2A Q03164 1/20 0.36
SLC6A2 P23975 1/20 0.36
SIGMAR1 Q99720 2/20 0.36
ADRA2A P08913 1/20 0.35
DRD2 P14416 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
DRD1 P21728 1/20 0.35
DRD5 P21918 1/20 0.35
DRD3 P35462 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
MAPK1 P28482 1/20 0.34
PRCP P42785 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1891904 0.73 SLC6A3 (0.44) PARP3SLC6A3SLC6A2CHRNB2CHRNA4
SCHEMBL612073 0.72 PDE4A (0.41) CYP3A4ADRA2ADRD2ADRA2BADRA2C
SCHEMBL2792608 0.71 MAOB (0.48) PARP3SLC6A3CYP3A4CYP2D6SLC6A2
SCHEMBL2790840 0.68 SLC6A3 (0.41) PARP3SLC6A3MTNR1ASIGMAR1
SCHEMBL10725693 0.68 MTNR1A (0.42) PARP3SLC6A3MTNR1AMEN1CYP3A4
SCHEMBL10720882 0.68 MTNR1A (0.42) PARP3SLC6A3MTNR1AMEN1CYP3A4
SCHEMBL10721311 0.68 MTNR1A (0.42) PARP3SLC6A3MTNR1AMEN1CYP3A4
SCHEMBL3150368 0.67 MAPK1 (0.56) MTNR1AMEN1KMT2AMAPK1
SCHEMBL3159001 0.67 MAPK1 (0.56) MTNR1AMEN1KMT2AMAPK1
SCHEMBL531338 0.67 MAPK1 (0.56) MTNR1AMEN1KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0201085-A2 6-Phenyl-1,2,3,4,4a,5,6,10b-octahydrobenz(h) isoquinolines PENNWALT CORPORATION (US) 1986-11-12 EP disclosed