SCHEMBL10876232

SCHEMBL10876232

Nc1nc2c(cc1F)c(=O)c(C(=O)O)cn2C1CC1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 6/20 0.59
CHRM2 P08172 2/20 0.54
DRD1 P21728 1/20 0.54
TOP2A P11388 8/20 0.53
TOP2B Q02880 8/20 0.53
DHFR P00374 1/20 0.51
KDM4E B2RXH2 4/20 0.50
ALDH1A1 P00352 4/20 0.50
LMNA P02545 3/20 0.50
HSD17B10 Q99714 3/20 0.50
HPGD P15428 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
ABCC4 O15439 1/20 0.50
POLB P06746 1/20 0.48
CHRM1 P11229 1/20 0.48
OPRM1 P35372 1/20 0.48
OPRD1 P41143 1/20 0.48
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5142702 0.88 DPP4 (0.58) DPP4CHRM2DRD1TOP2ATOP2B
SCHEMBL9437304 0.88 TOP2A (0.58) DPP4CHRM2DRD1TOP2ATOP2B
SCHEMBL500472 0.85 DPP4 (0.57) DPP4CHRM2DRD1TOP2ATOP2B
SCHEMBL10330767 0.85 TOP2A (0.59) DPP4CHRM2DRD1TOP2ATOP2B
SCHEMBL10876616 0.85 DPP4 (0.56) DPP4CHRM2DRD1TOP2ATOP2B
SCHEMBL10876239 0.85 DPP4 (0.45) DPP4CHRM2DRD1TOP2ATOP2B
SCHEMBL17537044 0.83 DPP4 (0.56) DPP4CHRM2DRD1TOP2ATOP2B
SCHEMBL14143514 0.82 DPP4 (0.54) DPP4CHRM2DRD1TOP2ATOP2B
SCHEMBL14472239 0.82 DPP4 (0.56) DPP4CHRM2DRD1TOP2ATOP2B
SCHEMBL10413901 0.82 DPP4 (0.55) DPP4CHRM2DRD1TOP2ATOP2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0203488-A2 7-Azolyl-1-cyclopropyl-1,4-dihydro-4-oxo-3-quinoline carboxylic acids and 1,8-naphthyridine carboxylic acids, process for their preparation and bactericidal agents containing them BAYER AG (DE) 1986-12-03 EP disclosed