SCHEMBL10878124

SCHEMBL10878124

Nc1ccccc1NS(=O)(=O)C1CCCC1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.50
GAA P10253 1/20 0.50
MAPT P10636 1/20 0.50
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.47
PGAM1 P18669 1/20 0.47
ACLY P53396 1/20 0.46
MRGPRX1 Q96LB2 5/20 0.44
ALOX5AP P20292 2/20 0.43
FEN1 P39748 2/20 0.43
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
BRD4 O60885 6/20 0.41
SGK1 O00141 1/20 0.39
CKS1B P61024 1/20 0.38
SKP2 Q13309 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20837041 0.98 KDM4E (0.53) KDM4EGAAMAPTHDAC3HDAC1
SCHEMBL22290162 0.93 PTGS1 (0.47) KDM4EGAAMAPTHDAC3HDAC1
SCHEMBL29739977 0.93 PTGS1 (0.47) KDM4EGAAMAPTHDAC3HDAC1
SCHEMBL23014676 0.74 ACLY (0.65) KDM4EGAAMAPTPGAM1ACLY
SCHEMBL23014672 0.74 PGAM1 (0.49) KDM4EPGAM1ACLYMRGPRX1PTGS1
SCHEMBL23014657 0.74 PGAM1 (0.46) KDM4EGAAPGAM1ACLYMRGPRX1
SCHEMBL13783840 0.74 HDAC1 (0.53) KDM4EGAAMAPTHDAC3HDAC1
SCHEMBL17404466 0.74 BRD4 (0.51) PGAM1ACLYPTGS1PTGS2BRD4
SCHEMBL449212 0.74 KEAP1 (0.55) KDM4EGAAMAPTPTGS1PTGS2
SCHEMBL29396266 0.74 KEAP1 (0.55) KDM4EGAAMAPTPTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0093591-B1 SELECTIVE SULFONATION PROCESS ELI LILLY AND COMPANY (US) 1986-01-15 EP disclosed
EP-0093591-A1 Selective sulfonation process ELI LILLY AND COMPANY (US) 1983-11-09 EP disclosed