SCHEMBL10885240

SCHEMBL10885240

Cc1c(N)cc(Cc2ccccc2N)cc1N

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.46
TSHR P16473 1/20 0.46
PIK3CA P42336 1/20 0.46
TDP1 Q9NUW8 1/20 0.43
ALDH1A1 P00352 2/20 0.39
SLC6A2 P23975 4/20 0.38
SLC6A4 P31645 4/20 0.38
TAAR1 Q96RJ0 1/20 0.38
SLC6A3 Q01959 1/20 0.37
CD44 P16070 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
AR P10275 1/20 0.37
ALOX15 P16050 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HTR2A P28223 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10799481 0.84 CYP3A4 (0.45) CYP3A4TSHRTDP1ALDH1A1TAAR1
SCHEMBL9800610 0.83 CYP3A4 (0.64) CYP3A4TSHRPIK3CATDP1ALDH1A1
SCHEMBL10510941 0.82 TDP1 (0.48) CYP3A4TDP1ALDH1A1SLC6A2SLC6A4
SCHEMBL10422322 0.81 CYP3A4 (0.50) CYP3A4TSHRPIK3CATDP1ALDH1A1
SCHEMBL12323449 0.81 PKM (0.46) CYP3A4TDP1ALDH1A1KDM4EHPGD
SCHEMBL11658684 0.79 POLB (0.44) CYP3A4TSHRTDP1ALDH1A1TAAR1
SCHEMBL10799437 0.79 SKP2 (0.49) CYP3A4TSHRTDP1ALDH1A1SLC6A2
SCHEMBL10805311 0.79 POLB (0.39) CYP3A4TDP1ALDH1A1SLC6A2SLC6A4
SCHEMBL6206260 0.78 CYP3A4 (0.52) CYP3A4TSHRTDP1ALDH1A1SLC6A2
SCHEMBL9493658 0.78 CALM1 (0.55) CYP3A4TSHRPIK3CAALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0027953-B2 PROCESS FOR PREPARING N,O-DISUBSTITUTED URETHANES BAYER AG (DE) 1986-11-05 EP disclosed
US-4430505-A UREA, PRIMARY AMINES, ALCOHOLS BAYER AKTIENGESELLSCHAFT (DE) 1984-02-07 US disclosed
EP-0027940-B1 PROCESS FOR PREPARING URETHANES BAYER AG (DE) 1983-09-14 EP disclosed
US-4388238-A FROM PRIMARY AMINES, ALCOHOLS, AND CARBONYL COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 1983-06-14 US disclosed
EP-0027952-B1 PROCESS FOR PREPARING N,O-DISUBSTITUTED URETHANES BAYER AG (DE) 1983-04-13 EP disclosed
EP-0027953-B1 PROCESS FOR PREPARING N,O-DISUBSTITUTED URETHANES BAYER AG (DE) 1983-02-16 EP disclosed
EP-0059400-A2 Process for the preparation of urethanes BAYER AG (DE) 1982-09-08 EP disclosed
EP-0027952-A1 Process for preparing N,O-disubstituted urethanes BAYER AG (DE) 1981-05-06 EP disclosed
EP-0027940-A1 Process for preparing urethanes BAYER AG (DE) 1981-05-06 EP disclosed
EP-0027953-A1 Process for preparing N,O-disubstituted urethanes BAYER AG (DE) 1981-05-06 EP disclosed