SCHEMBL10899448

SCHEMBL10899448

CC1N/C(=C\c2cccc(Oc3ccccc3)c2)C(=O)O1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 4/20 0.48
MMP3 P08254 2/20 0.46
MMP13 P45452 2/20 0.46
SIRT1 Q96EB6 1/20 0.44
PARP1 P09874 1/20 0.41
TLR4 O00206 1/20 0.41
TLR2 O60603 1/20 0.41
NTRK1 P04629 1/20 0.41
ADAMTS5 Q9UNA0 4/20 0.40
ALOX5 P09917 3/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
PSMB5 P28074 1/20 0.40
ALPI P09923 1/20 0.39
GPR18 Q14330 1/20 0.38
PTPN1 P18031 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10898759 0.84 AKR1B1 (0.51) AKR1B1MMP3MMP13SIRT1PARP1
SCHEMBL8958542 0.83 LMNA (0.43) SIRT1ALPI
SCHEMBL10897268 0.76 KMT2A (0.44) PTGS2
SCHEMBL8170053 0.75 RXRA (0.45) AKR1B1MMP3MMP13ADAMTS5
SCHEMBL10730264 0.74 AKR1B1 (0.49) AKR1B1MMP3MMP13PARP1TLR4
SCHEMBL10899305 0.73 DYRK1A (0.54) AKR1B1PSMB5ALPI
SCHEMBL10898779 0.73 KMT2A (0.55) PSMB5
SCHEMBL8961052 0.73 NOTUM (0.39) SIRT1
SCHEMBL8961053 0.73 NOTUM (0.39) SIRT1
SCHEMBL10900059 0.72 IGF1R (0.42) SIRT1ADAMTS5PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4612388-A Process for producing N-acylphenylalanines MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1986-09-16 US claimed
US-4612388-A Process for producing N-acylphenylalanines MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1986-09-16 US disclosed
EP-0161796-A1 Process for producing N-acylphenylalanines MITSUI TOATSU CHEMICALS, Inc. (JP) 1985-11-21 EP disclosed