SCHEMBL10903820

SCHEMBL10903820

Cc1nccn1-c1ccc(N)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.44
KDM4E B2RXH2 2/20 0.44
RAD52 P43351 1/20 0.44
ALDH1A1 P00352 4/20 0.44
POLB P06746 1/20 0.44
CYP3A4 P08684 4/20 0.43
HTT P42858 1/20 0.43
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NFKB1 P19838 1/20 0.40
PMP22 Q01453 1/20 0.40
CYP2E1 P05181 1/20 0.39
CYP2A6 P11509 1/20 0.39
KCNH2 Q12809 1/20 0.39
TSHR P16473 1/20 0.38
BDKRB2 P30411 1/20 0.37
KDR P35968 1/20 0.37
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3431048 0.81 NR3C2 (0.46) MAPTKDM4EALDH1A1CYP3A4CYP2E1
SCHEMBL15218939 0.78 NR4A1 (0.54) MAPTKDM4EALDH1A1CYP3A4HTT
SCHEMBL1926995 0.77 ALDH1A1 (0.49) MAPTKDM4EALDH1A1POLBCYP3A4
SCHEMBL12342913 0.76 CYP3A4 (0.47) KDM4EALDH1A1CYP3A4CYP2E1CYP2A6
SCHEMBL11624615 0.75 ADH5 (0.46) KDM4EALDH1A1CYP3A4CYP2E1CYP2A6
SCHEMBL27556239 0.74 CYP3A4 (0.39) ALDH1A1CYP3A4SMN1; SMN2CYP2E1CYP2A6
SCHEMBL3509305 0.72 ICMT (0.55) CYP3A4CYP2E1CYP2A6BDKRB2GRM5
SCHEMBL31253290 0.72 AHR (0.34) KDM4EALDH1A1CYP3A4CYP2E1CYP2A6
SCHEMBL265184 0.72 ALDH1A1 (0.61) MAPTALDH1A1CYP3A4GAACYP2E1
SCHEMBL19814656 0.71 MAPT (0.44) MAPTKDM4ERAD52ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4533669-A NONTOXIC EISAI CO., LTD. (JP) 1985-08-06 US claimed
US-4602031-A Anti-depressant imidazoles, compositions and use EISAI CO., LTD. (JP) 1986-07-22 US disclosed
US-4533669-A NONTOXIC EISAI CO., LTD. (JP) 1985-08-06 US disclosed
US-4402966-A Acylaminophenyl imidazoles and anti-depressing agent containing the same EISAI CO., LTD. (JP) 1983-09-06 US disclosed
US-4301169-A Novel imidazole compound and anti-depressing agent containing the same EISAI CO., LTD. (JP) 1981-11-17 US disclosed