SCHEMBL10923751

SCHEMBL10923751

Nc1nc(Cl)nc(-c2ccc(Cl)c(Cl)c2)n1

nearest known ligand 0.82

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.82
NPC1 O15118 2/20 0.82
HRH4 Q9H3N8 2/20 0.55
KMO O15229 3/20 0.49
DHFR P00374 1/20 0.47
AHR P35869 2/20 0.46
HTR2B P41595 1/20 0.44
PDE4D Q08499 1/20 0.44
IKBKB O14920 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ADORA1 P30542 1/20 0.42
CYP1B1 Q16678 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9566581 0.90 RAB9A (1.00) RAB9ANPC1HRH4KMODHFR
SCHEMBL10925902 0.79 NPC1 (0.80) RAB9ANPC1HRH4DHFRHTR2B
SCHEMBL9566548 0.77 RAB9A (0.75) RAB9ANPC1HRH4KMODHFR
SCHEMBL9566620 0.77 RAB9A (0.75) RAB9ANPC1HRH4DHFRHTR2B
SCHEMBL6584030 0.76 HRH4 (0.56) RAB9ANPC1HRH4DHFRADORA1
SCHEMBL6986219 0.76 ADORA1 (0.67) RAB9ANPC1HRH4IKBKBKDM4E
SCHEMBL27774680 0.76 NPC1 (0.57) RAB9ANPC1HRH4DHFRIKBKB
SCHEMBL10923642 0.75 RAB9A (0.64) RAB9ANPC1HRH4KMODHFR
SCHEMBL2250601 0.75 ADORA2A (0.72) RAB9ANPC1HRH4KDM4EALDH1A1
SCHEMBL30205277 0.75 ADORA2A (0.72) RAB9ANPC1HRH4KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015155129-A1 DIAMINOTRIAZINE COMPOUND BASF SE (DE) 2015-10-15 WO disclosed
EP-0066799-B1 NICOTINIC ACID DERIVATIVES NIPPON SHINYAKU COMPANY, LIMITED (JP) 1986-01-02 EP disclosed
US-4415570-A TREATMENT FOR RHEMATIC DISEASES AND ALLERGIC NEPHRYTIS; UROGENITAL DISORDERS NIPPON SHINYAKU CO. LTD. (JP) 1983-11-15 US disclosed
EP-0066799-A2 Nicotinic acid derivatives NIPPON SHINYAKU COMPANY, LIMITED (JP) 1982-12-15 EP disclosed
US-4333933-A ANTIINFLAMMATORY, REACTING HALO BENZOGUANAMINE WITH NICOTINE ACID DERIVAGIVE NIPPON SHINYAKU CO., LTD. (JP) 1982-06-08 US disclosed