SCHEMBL10948840

SCHEMBL10948840

CN(C)CCOc1cccc(OCCCN)c1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.63
CHRNA4 P43681 3/20 0.63
KEAP1 Q14145 1/20 0.57
NFE2L2 Q16236 1/20 0.57
KDM4E B2RXH2 6/20 0.54
ALDH1A1 P00352 4/20 0.54
LMNA P02545 1/20 0.54
LTA4H P09960 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.52
NOS1 P29475 2/20 0.51
NOS2 P35228 2/20 0.51
ESR1 P03372 1/20 0.49
NOS3 P29474 1/20 0.49
MAPT P10636 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10950517 0.84 ACHE (0.54) CHRNB2CHRNA4KEAP1NFE2L2NOS1
SCHEMBL10955368 0.83 NOS1 (0.55) CHRNB2CHRNA4KEAP1NFE2L2KDM4E
SCHEMBL30862627 0.82 CHRNB2 (0.67) CHRNB2CHRNA4KEAP1NFE2L2KDM4E
SCHEMBL5025139 0.82 CHRNB2 (0.67) CHRNB2CHRNA4KEAP1NFE2L2KDM4E
SCHEMBL16858365 0.82 CHRNB2 (0.67) CHRNB2CHRNA4KEAP1NFE2L2KDM4E
SCHEMBL26995599 0.82 TAAR1 (0.58) CHRNB2CHRNA4KEAP1NFE2L2KDM4E
SCHEMBL781665 0.81 KEAP1 (0.70) CHRNB2CHRNA4KEAP1NFE2L2KDM4E
SCHEMBL1641682 0.81 CHRNB2 (0.65) CHRNB2CHRNA4KEAP1NFE2L2KDM4E
SCHEMBL11934997 0.80 CHRNB2 (0.49) CHRNB2CHRNA4KEAP1NFE2L2KDM4E
SCHEMBL16718937 0.80 MAPK1 (0.59) ALDH1A1LMNASMN1; SMN2NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4496567-A HSITAMINE H2 ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1985-01-29 US disclosed
EP-0013071-A1 Pyrimidinone derivatives, processes for preparing them and pharmaceutical compositions containing them SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1980-07-09 EP disclosed
WO-1980000966-A1 NEW HISTAMINE H2-ANTAGONISTS SMITH KLINE FRENCH LAB (GB) 1980-05-15 WO disclosed