SCHEMBL10956169

SCHEMBL10956169

NC(=S)/C=C(/N)c1ccc(Cl)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.45
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
POLB P06746 1/20 0.38
TSHR P16473 3/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
ALOX15 P16050 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPK1 P28482 1/20 0.38
ATM Q13315 1/20 0.38
ALDH1A1 P00352 3/20 0.38
MAPT P10636 3/20 0.38
KDM4E B2RXH2 2/20 0.38
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
EGFR P00533 1/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
PHGDH O43175 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10956171 1.00 LMNA (0.45) LMNACES2CES1POLBTSHR
SCHEMBL12714065 0.78 CES2 (0.50) LMNACES2CES1TSHRL3MBTL1
SCHEMBL11124456 0.78 METTL3 (0.42) CES2CES1ATMALDH1A1MAPT
SCHEMBL11124453 0.78 METTL3 (0.42) CES2CES1ATMALDH1A1MAPT
SCHEMBL1838629 0.78 TSHR (0.44) TSHRMAPTEGFRPHGDHSMN1; SMN2
SCHEMBL1838631 0.78 TSHR (0.44) TSHRMAPTEGFRPHGDHSMN1; SMN2
SCHEMBL12285402 0.77 MAPT (0.42) POLBTSHRL3MBTL1CYP3A4ATM
SCHEMBL1839901 0.77 MAPT (0.42) POLBTSHRL3MBTL1CYP3A4ATM
SCHEMBL1839902 0.77 MAPT (0.42) POLBTSHRL3MBTL1CYP3A4ATM
SCHEMBL6662812 0.77 ALOX15 (0.52) LMNACES2CES1TSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0135252-A2 Process for preparing 3-substituted-3-aminonitrile ELI LILLY AND COMPANY (US) 1985-03-27 EP disclosed
EP-0129407-A2 Improvements in and relating to (3-aryl-5-isothiazolyl)ureas ELI LILLY AND COMPANY (US) 1984-12-27 EP disclosed