SCHEMBL10974445

SCHEMBL10974445

CC(=O)OC(C)(C(=O)Nc1ccc(C#N)c(C#N)c1)C(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
ABCC9 O60706 3/20 0.47
ABCC8 Q09428 3/20 0.47
KCNJ11 Q14654 3/20 0.47
KCNJ8 Q15842 3/20 0.47
AR P10275 4/20 0.44
PDK1 Q15118 1/20 0.43
PDK2 Q15119 1/20 0.43
PDK3 Q15120 1/20 0.43
PDK4 Q16654 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8518923 0.84 ALDH1A1 (0.55) ALDH1A1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL7515733 0.80 ABCC9 (0.68) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL8519769 0.77 ALDH1A1 (0.54) ALDH1A1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8519617 0.76 ALDH1A1 (0.57) ALDH1A1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL14087515 0.74 ALDH1A1 (0.55) ALDH1A1AR
SCHEMBL8983980 0.74 ALDH1A1 (0.70) ALDH1A1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL10984365 0.74 AR (0.54) ARCYP2C19
SCHEMBL8351343 0.73 ALDH1A1 (0.79) ALDH1A1CYP2C19
SCHEMBL10976571 0.71 AR (0.69) ALDH1A1ARCYP2C19
SCHEMBL11226270 0.71 ALDH1A1 (0.43) ALDH1A1ABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0002892-B1 AMIDE DERIVATIVES, PROCESS FOR THEIR MANUFACTURE AND PHARMACEUTICAL OR VETERINARY COMPOSITIONS CONTAINING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-02-06 EP disclosed
US-4191775-A ANTIANDROGENIC IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1980-03-04 US disclosed
EP-0002892-A1 Amide derivatives, process for their manufacture and pharmaceutical or veterinary compositions containing them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1979-07-11 EP disclosed