SCHEMBL8518923

SCHEMBL8518923

CC(=O)OC(C)(C)C(=O)Nc1ccc(C#N)c(C#N)c1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.55
ABCC9 O60706 3/20 0.46
ABCC8 Q09428 3/20 0.46
KCNJ11 Q14654 3/20 0.46
KCNJ8 Q15842 3/20 0.46
AR P10275 5/20 0.44
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8519617 0.86 ALDH1A1 (0.57) ALDH1A1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL10974445 0.84 ALDH1A1 (0.50) ALDH1A1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8519769 0.81 ALDH1A1 (0.54) ALDH1A1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL11226270 0.80 ALDH1A1 (0.43) ALDH1A1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL11224840 0.80 ALDH1A1 (0.43) ALDH1A1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL14087515 0.78 ALDH1A1 (0.55) ALDH1A1AR
SCHEMBL8351343 0.77 ALDH1A1 (0.79) ALDH1A1CYP2C19
SCHEMBL7515733 0.76 ABCC9 (0.68) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL10984365 0.75 AR (0.54) ARCYP2C19
SCHEMBL5199230 0.74 L3MBTL1 (0.46) ALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5994362-A ADMINISTERING FINASTERIDE AND CASODEX MERCK & CO., INC. (US) 1999-11-30 US disclosed
EP-0514056-A2 Use of estrogens or antiandrogens for reversal of male sexual phenotype in poultry MERCK & CO. INC. (US) 1992-11-19 EP disclosed
WO-1992016233-A1 PHARMACEUTICAL COMBINATION FOR THE TREATMENT OF PROSTATIC CANCER CONTAINING A 5 ALPHA REDUCTASE INHIBITOR AND AN ANTIANDROGEN MERCK & CO., INC. (US) 1992-10-01 WO disclosed
EP-0002309-B1 ACYLANILIDES, PROCESS FOR THEIR MANUFACTURE AND PHARMACEUTICAL AND VETERINARY COMPOSITIONS CONTAINING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-12-01 EP disclosed
US-4282218-A ANTIANDROGENS IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1981-08-04 US disclosed
US-4239776-A Anti-androgenic amides IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1980-12-16 US disclosed
EP-0002309-A2 Acylanilides, process for their manufacture and pharmaceutical and veterinary compositions containing them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1979-06-13 EP disclosed