SCHEMBL10976089

SCHEMBL10976089

Clc1ccc2cc(Cl)ncc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.50
NOS1 P29475 2/20 0.41
NR4A2 P43354 2/20 0.41
DYRK1A Q13627 1/20 0.41
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
NPC1 O15118 1/20 0.38
CHEK1 O14757 1/20 0.37
HTR3A P46098 1/20 0.37
F11 P03951 1/20 0.35
AHR P35869 2/20 0.34
CMA1 P23946 1/20 0.34
F7 P08709 1/20 0.34
LTA4H P09960 1/20 0.34
F3 P13726 1/20 0.34
ABL1 P00519 3/20 0.33
GRM4 Q14833 1/20 0.33
TP53 P04637 1/20 0.33
CDC7 O00311 1/20 0.33
CDK2 P24941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2749728 0.78 CYP2A6 (0.46) CYP2A6NOS1NR4A2DYRK1APDGFRB
SCHEMBL14330642 0.78 CYP2A6 (0.46) CYP2A6NOS1NR4A2DYRK1APDGFRB
SCHEMBL4386257 0.78 CYP2A6 (0.57) CYP2A6NOS1NR4A2DYRK1AHTR3A
SCHEMBL558994 0.78 PDPK1 (0.57) CYP2A6NOS1NR4A2DYRK1ALTA4H
SCHEMBL933672 0.78 CYP2A6 (0.46) CYP2A6NOS1DYRK1AABL1GRM4
SCHEMBL8268451 0.78 CYP1A2 (0.54) CYP2A6ABL1
SCHEMBL10024955 0.78 ALDH1A1 (0.46) GRM4TP53CDC7CDK2
SCHEMBL17336629 0.78 NOS1 (0.38) NOS1NPC1ABL1GRM4CDC7
SCHEMBL10978740 0.78 L3MBTL1 (0.50) CYP2A6PDGFRBPDGFRAABL1
SCHEMBL16295919 0.78 CYP1A2 (0.46) ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103562199-B As the tripeptides mixing deuterium of hepatitis C virus inhibitors BRISTOL-MYERS SQUIBB CO. (US) 2016-03-30 CN disclosed
CN-103562199-A Tripeptides incorporating deuterium as inhibitors of hepatitis c virus BRISTOL MYERS SQUIBB CO 2014-02-05 CN disclosed
EP-0048539-B1 ISOQUINOLYLOXY(AMINO)PHENOXYALKANE CARBOXYLIC ACID DERIVATIVES, PROCESS FOR THEIR SYNTHESIS, HERBICIDAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS HERBICIDES ICI AUSTRALIA LIMITED (AU) 1985-08-28 EP disclosed
US-4409017-A Herbicidal isoquinolinoxy- or isoquinolinamino-phenoxy alkane carboxylic acid derivatives ICI AUSTRALIA LIMITED (AU) 1983-10-11 US disclosed
EP-0048539-A1 Isoquinolyloxy(amino)phenoxyalkane carboxylic acid derivatives, process for their synthesis, herbicidal compositions containing them and their use as herbicides ICI AUSTRALIA LIMITED (AU) 1982-03-31 EP disclosed