SCHEMBL10979871

SCHEMBL10979871

O=c1[nH]c(=O)c2nc(-c3ccccc3)c(-c3ccccc3)nc2[nH]1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 1/20 0.68
KDM4E B2RXH2 6/20 0.62
ALDH1A1 P00352 5/20 0.62
HSD17B10 Q99714 3/20 0.62
ADORA2A P29274 3/20 0.62
RAB9A P51151 3/20 0.62
BLM P54132 2/20 0.62
TDP1 Q9NUW8 2/20 0.62
ADORA2B P29275 2/20 0.62
CYP1A2 P05177 1/20 0.62
PABPC1 P11940 1/20 0.62
CYP2C19 P33261 1/20 0.62
CASP7 P55210 1/20 0.62
PMP22 Q01453 1/20 0.62
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
POLB P06746 2/20 0.58
LMNA P02545 1/20 0.58
MAPT P10636 1/20 0.58
PKM P14618 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7833902 0.87 KDM4E (0.55) PIK3CGKDM4EALDH1A1HSD17B10ADORA2A
SCHEMBL20798351 0.83 XDH (0.55) PIK3CGKDM4EALDH1A1HSD17B10ADORA2A
SCHEMBL29467240 0.83 XDH (0.55) PIK3CGKDM4EALDH1A1HSD17B10ADORA2A
SCHEMBL31214529 0.81 ALDH1A1 (0.60) PIK3CGKDM4EALDH1A1HSD17B10ADORA2A
Alloxazine SCHEMBL499075 0.77 KDM4E (1.00) PIK3CGKDM4EALDH1A1HSD17B10ADORA2A
Alloxazine SCHEMBL29516835 0.77 KDM4E (1.00) PIK3CGKDM4EALDH1A1HSD17B10ADORA2A
SCHEMBL10983379 0.76 KDM4E (0.74) PIK3CGKDM4EALDH1A1HSD17B10ADORA2A
SCHEMBL3225296 0.76 KDM4E (0.74) PIK3CGKDM4EALDH1A1HSD17B10ADORA2A
SCHEMBL824381 0.76 PIK3CG (0.56) PIK3CGKDM4EALDH1A1HSD17B10ADORA2A
SCHEMBL11087373 0.75 KDM4E (0.69) PIK3CGKDM4EALDH1A1HSD17B10ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071903-B1 DIGLYCIDYL PTERIDINE COMPOUNDS, METHOD FOR THEIR PREPARATION AND THEIR USE IN DRUGS WITH A CYTOSTATIC ACTIVITY Henkel Kommanditgesellschaft auf Aktien (DE) 1985-08-28 EP disclosed
US-4463006-A ANTICANCER, ANTITUMOR AGENTS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1984-07-31 US disclosed
EP-0071903-A1 Diglycidyl pteridine compounds, method for their preparation and their use in drugs with a cytostatic activity Henkel Kommanditgesellschaft auf Aktien (DE) 1983-02-16 EP disclosed