SCHEMBL10980261

SCHEMBL10980261

CC(Br)c1cccc(Cl)c1Cl

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.63
PNMT P11086 2/20 0.63
CYP3A4 P08684 2/20 0.63
CYP2D6 P10635 1/20 0.63
NFKB1 P19838 1/20 0.63
LMNA P02545 3/20 0.61
ALDH1A1 P00352 1/20 0.61
GLA P06280 1/20 0.61
P2RX7 Q99572 1/20 0.58
IDO1 P14902 1/20 0.42
TDO2 P48775 1/20 0.42
TSHR P16473 4/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35
KCNH2 Q12809 1/20 0.35
CYP2A6 P11509 1/20 0.35
FAAH O00519 1/20 0.34
CA1 P00915 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL320794 0.81 P2RX7 (0.47) CYP1A2PNMTCYP3A4CYP2D6NFKB1
SCHEMBL13145151 0.81 P2RX7 (0.47) CYP1A2PNMTCYP3A4CYP2D6NFKB1
SCHEMBL423182 0.81 CYP1A2 (0.68) CYP1A2PNMTCYP3A4CYP2D6NFKB1
SCHEMBL22801396 0.81 CYP1A2 (0.68) CYP1A2PNMTCYP3A4CYP2D6NFKB1
SCHEMBL11499495 0.81 CYP1A2 (0.56) CYP1A2PNMTCYP3A4CYP2D6NFKB1
SCHEMBL25392757 0.80 P2RX7 (0.56) CYP1A2PNMTCYP3A4CYP2D6NFKB1
SCHEMBL1281895 0.80 P2RX7 (0.47) CYP1A2PNMTCYP3A4CYP2D6NFKB1
SCHEMBL30785267 0.80 P2RX7 (0.56) CYP1A2PNMTCYP3A4CYP2D6NFKB1
SCHEMBL8440315 0.79 P2RX7 (0.46) CYP1A2PNMTCYP3A4CYP2D6NFKB1
SCHEMBL11501928 0.79 CYP1A2 (0.65) CYP1A2PNMTCYP3A4CYP2D6NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0159915-A2 Process for making ring-halogenated styrenes and their use YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 1985-10-30 EP claimed
CN-102666545-B As the heterocycle Pyrazolopyrimidine analogs of JAK inhibitor CELLZOME LTD. (GB) 2016-04-06 CN disclosed
CN-104395310-A Bicyclic substituted uracils and their use Bayer Pharma AG 2015-03-04 CN disclosed
CN-104039791-A [1,2,3] triazolo [4,5-D ] pyrimidine derivatives as cannabinoid receptor 2 agonists HOFFMANN LA ROCHE 2014-09-10 CN disclosed
CN-103930426-A [1, 2, 3] triazolo [4, 5 -d] pyrimidine derivatives as agonists of the cannabinoid receptor 2 HOFFMANN LA ROCHE 2014-07-16 CN disclosed
EP-0159915-A2 Process for making ring-halogenated styrenes and their use YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 1985-10-30 EP disclosed