SCHEMBL10994657

SCHEMBL10994657

Cc1ccc2c(c1)OCC(C(O)CN1CCN(C(C(N)=O)c3ccc(C(F)(F)F)cc3)CC1)O2

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TEAD1 P28347 6/20 0.42
CYP2D6 P10635 6/20 0.38
OGA O60502 2/20 0.34
MC4R P32245 1/20 0.34
CCR3 P51677 1/20 0.33
FFAR1 O14842 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10995105 0.92 CYP2D6 (0.35) CYP2D6FFAR1
SCHEMBL10995041 0.89 ALDH1A1 (0.36) CYP2D6
SCHEMBL10996165 0.89 TEAD1 (0.42) TEAD1CYP2D6
SCHEMBL7436237 0.86 TEAD1 (0.42) TEAD1OGACCR3
SCHEMBL10991901 0.84 LMNA (0.42) CYP2D6
SCHEMBL10994531 0.83 CA2 (0.34) CYP2D6
SCHEMBL10993606 0.83 TEAD1 (0.35) TEAD1CYP2D6FFAR1
SCHEMBL10997571 0.83 FFAR1 (0.34) CYP2D6FFAR1
SCHEMBL10993683 0.82 ALDH1A1 (0.37) OGAMC4RFFAR1
SCHEMBL10991654 0.81 CHRM2 (0.43) CYP2D6FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4558129-A Benzodioxanyl-hydroxyethylene-piperazinyl acetanilides which effect calcium entry and β-blockade SYNTEX (U.S.A.) INC. (US) 1985-12-10 US disclosed