SCHEMBL11005353

SCHEMBL11005353

COC(=O)c1cc(Cc2ccc(OC)cc2)ns1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SAE1 Q9UBE0 1/20 0.46
UBA2 Q9UBT2 1/20 0.46
OPRD1 P41143 1/20 0.44
ALDH1A1 P00352 3/20 0.43
LMNA P02545 2/20 0.43
MAPT P10636 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
HTT P42858 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP1A2 P05177 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP2D6 P10635 1/20 0.41
TP53 P04637 2/20 0.41
F2RL1 P55085 1/20 0.41
GAA P10253 1/20 0.41
ALOX12 P18054 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11000260 0.90 KDM5A (0.45) SAE1UBA2ALDH1A1LMNAMAPT
SCHEMBL11004923 0.85 PRKACA (0.45) ALDH1A1MAPTHTTMEN1KMT2A
SCHEMBL11001932 0.76 KDM4C (0.48) ALDH1A1HTTMEN1KMT2ACYP1A2
SCHEMBL11005342 0.75 MAPT (0.54) OPRD1ALDH1A1LMNAMAPTCA1
SCHEMBL19844014 0.71 KDM4E (0.56) SAE1UBA2ALDH1A1MAPTCA1
SCHEMBL8993003 0.71 CA1 (0.78) SAE1UBA2ALDH1A1LMNAMAPT
SCHEMBL95380 0.70 HPGD (0.56) SAE1UBA2ALDH1A1LMNAMAPT
SCHEMBL15831652 0.70 ALDH1A1 (0.56) SAE1UBA2ALDH1A1LMNAMAPT
SCHEMBL13539015 0.70 KDM4E (0.56) SAE1UBA2ALDH1A1LMNAMAPT
SCHEMBL27643975 0.69 MAPT (0.49) SAE1UBA2ALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4544752-A TREATMENT OF GOUT; ANTIARTHRITIC AGENTS ELI LILLY AND COMPANY (US) 1985-10-01 US disclosed
US-4346094-A ENZYME INHIBITORS ELI LILLY AND COMPANY (US) 1982-08-24 US disclosed
EP-0048615-A1 Improvements in or relating to 3-aryl-5-isothiazole derivatives ELI LILLY AND COMPANY (US) 1982-03-31 EP disclosed