SCHEMBL11010378

SCHEMBL11010378

COc1cc(NC(C)C#N)ccc1-c1nc2cncnc2[nH]1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 13/20 0.39
AAK1 Q2M2I8 3/20 0.36
PDE5A O76074 2/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
EGFR P00533 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11010396 0.85 ENPP1 (0.42) CYP17A1AAK1PDE5APDE3BPDE3A
SCHEMBL11010174 0.83 CYP17A1 (0.39) CYP17A1AAK1PDE5APDE3BPDE3A
SCHEMBL11010226 0.83 AAK1 (0.42) CYP17A1AAK1PDE5APDE3BPDE3A
SCHEMBL11007244 0.82 PDE2A (0.38) CYP17A1AAK1PDE5APDE3BPDE3A
SCHEMBL11005537 0.79 CYP17A1 (0.39) CYP17A1AAK1PDE5APDE3BPDE3A
SCHEMBL11237399 0.78 PDE2A (0.51) CYP17A1PDE5APDE3BPDE3AEGFR
SCHEMBL11011297 0.78 IMPDH2 (0.45) PDE5APDE3BPDE3AEGFR
SCHEMBL11008020 0.77 PDE2A (0.39) PDE5APDE3BPDE3AEGFR
SCHEMBL11356780 0.77 AMY1A (0.47) CYP17A1PDE5APDE3BPDE3A
SCHEMBL11006162 0.77 CDK4 (0.43) PDE5APDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142075-A2 Purine derivatives, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-05-22 EP disclosed