SCHEMBL11014756

SCHEMBL11014756

CCOC(=O)Nc1c(Cl)cc(Cl)cc1C(=O)OCC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
ABCB1 P08183 1/20 0.49
NLRP3 Q96P20 1/20 0.46
MAPT P10636 2/20 0.45
KDM4E B2RXH2 4/20 0.44
HPGD P15428 3/20 0.44
GAA P10253 2/20 0.44
GLA P06280 1/20 0.44
CYP4F2 P78329 1/20 0.43
CYP4A11 Q02928 1/20 0.43
BAZ2B Q9UIF8 1/20 0.43
BAZ2A Q9UIF9 1/20 0.43
ALOX15 P16050 1/20 0.43
KMT2A Q03164 2/20 0.43
TP53 P04637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA7 P43166 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11867300 0.82 ABCB1 (0.51) ALDH1A1ABCB1NLRP3MAPTKDM4E
SCHEMBL30201359 0.77 NLRP3 (0.48) ALDH1A1ABCB1NLRP3MAPTKDM4E
SCHEMBL1096330 0.77 NLRP3 (0.48) ALDH1A1ABCB1NLRP3MAPTKDM4E
SCHEMBL11682561 0.76 AKR1C4 (0.55) ALDH1A1MAPTKDM4EHPGDGAA
SCHEMBL9268795 0.76 ABCB1 (0.48) ALDH1A1ABCB1MAPTKDM4ECYP4F2
SCHEMBL9727774 0.75 ALDH1A1 (0.71) ALDH1A1MAPTKDM4EHPGDGAA
SCHEMBL7558526 0.75 NLRP3 (0.54) ALDH1A1ABCB1NLRP3KDM4EGLA
SCHEMBL11545231 0.74 NLRP3 (0.52) ALDH1A1ABCB1NLRP3MAPTKDM4E
SCHEMBL14489629 0.74 KDM4E (0.50) ALDH1A1NLRP3MAPTKDM4EHPGD
SCHEMBL11010057 0.73 ALDH1A1 (0.56) ALDH1A1KDM4EHPGDALOX15KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4522945-A SEROTONINE ANTAGONISTS JANSSEN PHARMACEUTICA N.V. (BE) 1985-06-11 US disclosed
EP-0013612-B1 (PIPERIDINYLALKYL)QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM JANSSEN PHARMACEUTICA N.V. (BE) 1983-11-09 EP disclosed
US-4335127-A POTENT SEROTONIN ANTAGONISTS JANSSEN PHARMACEUTICA, N.V. (BE) 1982-06-15 US disclosed
EP-0013612-A2 (Piperidinylalkyl)quinazoline derivatives, process for their preparation and pharmaceutical compositions containing them JANSSEN PHARMACEUTICA N.V. (BE) 1980-07-23 EP disclosed