SCHEMBL9727774

SCHEMBL9727774

CCOC(=O)c1cc(Cl)cc(Cl)c1N

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 13/20 0.71
KDM4E B2RXH2 12/20 0.71
GAA P10253 11/20 0.71
HPGD P15428 9/20 0.71
GLA P06280 8/20 0.71
NPSR1 Q6W5P4 1/20 0.68
SMN1; SMN2 Q16637 2/20 0.59
MAPT P10636 2/20 0.59
HSD17B10 Q99714 2/20 0.59
POLB P06746 2/20 0.57
ESR2 Q92731 1/20 0.57
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
PKM P14618 1/20 0.51
CTDSP1 Q9GZU7 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
MAPK1 P28482 1/20 0.50
CYP4F2 P78329 1/20 0.48
CYP4A11 Q02928 1/20 0.48
BAZ2B Q9UIF8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11025131 0.87 ALDH1A1 (0.66) ALDH1A1KDM4EGAAHPGDGLA
SCHEMBL16529438 0.87 ALDH1A1 (0.55) ALDH1A1KDM4EGAAHPGDGLA
SCHEMBL6948296 0.87 ALDH1A1 (0.55) ALDH1A1KDM4EGAAHPGDGLA
SCHEMBL29264039 0.85 ALDH1A1 (0.54) ALDH1A1KDM4EGAAHPGDGLA
SCHEMBL5409626 0.85 ALDH1A1 (0.54) ALDH1A1KDM4EGAAHPGDGLA
SCHEMBL28825145 0.84 ALDH1A1 (0.53) ALDH1A1KDM4EGAAHPGDGLA
SCHEMBL3585477 0.84 ALDH1A1 (0.52) ALDH1A1KDM4EGAAHPGDGLA
SCHEMBL30361197 0.83 CA1 (0.52) ALDH1A1KDM4EGAAHPGDGLA
SCHEMBL26466636 0.83 CA1 (0.52) ALDH1A1KDM4EGAAHPGDGLA
SCHEMBL11682561 0.81 AKR1C4 (0.55) ALDH1A1KDM4EGAAHPGDGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2754651-B1 NITROBENZENE COMPOUND MANUFACTURING METHOD KUMIAI CHEMICAL INDUSTRY CO (JP) 2017-12-06 EP disclosed
US-9006477-B2 Method for producing nitrobenzene compound IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2015-04-14 US disclosed
US-20140163256-A1 METHOD FOR PRODUCING NITROBENZENE COMPOUND IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2014-06-12 US disclosed
US-5132314-A For administration to mammals, anthranilic acid derivatives CIBA-GEIGY CORPORATION (US) 1992-07-21 US disclosed
US-5081125-A Substituted anthranilic acid derivatives CIBA-GEIGY CORPORATION (US) 1992-01-14 US disclosed
EP-0420804-A2 Anthelmintic compounds CIBA-GEIGY AG (CH) 1991-04-03 EP disclosed
EP-0101330-B1 2-QUINOLONE DERIVATIVES NIPPON SHINYAKU COMPANY, LIMITED (JP) 1988-08-24 EP disclosed
US-4526894-A Antiinflammatory agents NIPPON SHINYAKU CO. LTD. (JP) 1985-07-02 US disclosed
US-4522945-A SEROTONINE ANTAGONISTS JANSSEN PHARMACEUTICA N.V. (BE) 1985-06-11 US disclosed
EP-0101330-A2 2-Quinolone derivatives NIPPON SHINYAKU COMPANY, LIMITED (JP) 1984-02-22 EP disclosed
EP-0013612-B1 (PIPERIDINYLALKYL)QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM JANSSEN PHARMACEUTICA N.V. (BE) 1983-11-09 EP disclosed
US-4335127-A POTENT SEROTONIN ANTAGONISTS JANSSEN PHARMACEUTICA, N.V. (BE) 1982-06-15 US disclosed
EP-0013612-A2 (Piperidinylalkyl)quinazoline derivatives, process for their preparation and pharmaceutical compositions containing them JANSSEN PHARMACEUTICA N.V. (BE) 1980-07-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140163256-A1 METHOD FOR PRODUCING NITROBENZENE COMPOUND NOX1, NOS2, CYB5R3 ALDH1A1 548/4885KDM4E 3790/4885GAA 2092/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.