SCHEMBL11019652

SCHEMBL11019652

CCSc1ccc(-c2nc3ccc(C(=O)OC)cc3[nH]2)c(OC)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 4/20 0.52
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
HTT P42858 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
HDAC6 Q9UBN7 3/20 0.48
BRD4 O60885 1/20 0.48
MMP2 P08253 1/20 0.47
MMP9 P14780 1/20 0.47
MMP8 P22894 1/20 0.47
MMP13 P45452 1/20 0.47
PKN1 Q16512 1/20 0.45
PKN2 Q16513 1/20 0.45
AMY1A P0DUB6 1/20 0.45
SIRT2 Q8IXJ6 3/20 0.44
SIRT1 Q96EB6 2/20 0.44
SIRT3 Q9NTG7 1/20 0.44
CYP2C9 P11712 1/20 0.44
ATM Q13315 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11019650 0.92 CHEK2 (0.43) CHEK2KDM4EALDH1A1LMNAHTT
SCHEMBL11017902 0.91 CHEK2 (0.53) CHEK2L3MBTL1HDAC6AMY1APDE4A
SCHEMBL11016463 0.90 CHEK2 (0.66) CHEK2
SCHEMBL11019907 0.89 CHEK2 (0.53) CHEK2KDM4EALDH1A1LMNAHTT
SCHEMBL11020867 0.84 TP53 (0.51) CHEK2KDM4EALDH1A1LMNAHTT
SCHEMBL11017897 0.82 PDE4A (0.44) CHEK2L3MBTL1AMY1APDE4APDE4B
SCHEMBL11016890 0.82 CHEK2 (0.63) CHEK2LMNA
SCHEMBL11016458 0.82 CHEK2 (0.55) CHEK2
SCHEMBL11019275 0.81 CHEK2 (0.48) CHEK2KDM4ELMNAHDAC6PKN1
SCHEMBL10760161 0.80 RHEB (0.47) CHEK2KDM4EALDH1A1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP disclosed