SCHEMBL11025403

SCHEMBL11025403

COC(=O)[C@@H](O)[C@@H](Cc1ccccc1)NC(=O)CNC(C)=O

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PYGL P06737 1/20 0.48
ATM Q13315 2/20 0.46
LTA4H P09960 1/20 0.44
POLB P06746 1/20 0.44
KLK5 Q9Y337 2/20 0.44
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44
TRPM8 Q7Z2W7 1/20 0.44
REN P00797 1/20 0.42
CTRB1 P17538 1/20 0.42
ALDH1A1 P00352 1/20 0.42
THRB P10828 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HSD17B10 Q99714 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11028602 0.88 MTNR1A (0.47) PYGLMTNR1AMTNR1BCTRB1
SCHEMBL11089192 0.88 MTNR1A (0.47) PYGLMTNR1AMTNR1BCTRB1
SCHEMBL11026867 0.86 MTNR1A (0.45) PYGLMTNR1AMTNR1BCTRB1
SCHEMBL11030131 0.84 MTNR1A (0.43) POLBMTNR1AMTNR1BCTRB1
Hydrochloric Acid SCHEMBL11026585 0.82 LTA4H (0.52) PYGLATMLTA4HPOLBKLK5
SCHEMBL22886596 0.78 LTA4H (0.52) PYGLATMLTA4HPOLBKLK5
SCHEMBL19258128 0.78 LTA4H (0.52) PYGLATMLTA4HPOLBKLK5
SCHEMBL7418811 0.77 TRPM8 (0.69) PYGLATMLTA4HTRPM8CTRB1
SCHEMBL5652568 0.77 TRPM8 (0.55) PYGLATMLTA4HPOLBKLK5
SCHEMBL8163494 0.77 TRPM8 (0.69) PYGLATMLTA4HTRPM8CTRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0077274-B1 3-AMINO-2-HYDROXY-4-PHENYLBUTANOIC ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1985-08-28 EP claimed
EP-0077274-A1 3-Amino-2-hydroxy-4-phenylbutanoic acid derivatives and pharmaceutical composition containing the same ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1983-04-20 EP claimed
US-4474764-A ANALGESICS ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1984-10-02 US disclosed