SCHEMBL11027618

SCHEMBL11027618

O=C1NCC(CCc2ccccc2)N(C(=O)c2ccccc2)C1=O

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.45
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
POLB P06746 1/20 0.41
SLC18A2 Q05940 1/20 0.40
ABCB1 P08183 1/20 0.40
FAAH O00519 1/20 0.39
SIGMAR1 Q99720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11028695 0.92 KCNH2 (0.39) KCNH2MEN1KMT2AFAAH
SCHEMBL11029433 0.84 SLC18A2 (0.43) KCNH2SLC18A2
SCHEMBL14687476 0.67 ACHE (0.46) MEN1KMT2APOLBSIGMAR1
SCHEMBL11031319 0.66 SLC18A2 (0.42) SLC18A2
SCHEMBL11025726 0.65 TACR2 (0.44)
SCHEMBL11026816 0.65 KMT2A (0.46) KCNH2MEN1KMT2AFAAH
SCHEMBL11288045 0.65 ATM (0.51) SLC18A2
SCHEMBL28328103 0.64 ABCB1 (0.60) KCNH2SLC18A2ABCB1
SCHEMBL1190776 0.62 CA1 (0.48) KMT2A
SCHEMBL1191156 0.62 CA1 (0.48) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0086678-B1 PROCESS FOR THE PREPARATION OF 2-ACYL-1,3,4,6,7,11B-2H-HEXAHYDRO-4-PYRAZINO(2,1-A)ISOQUINOLINONES AND INTERMEDIATES ELF SANOFI (FR) 1985-07-03 EP claimed
EP-0086678-B1 PROCESS FOR THE PREPARATION OF 2-ACYL-1,3,4,6,7,11B-2H-HEXAHYDRO-4-PYRAZINO(2,1-A)ISOQUINOLINONES AND INTERMEDIATES ELF SANOFI (FR) 1985-07-03 EP disclosed
EP-0086678-A1 Process for the preparation of 2-acyl-1,3,4,6,7,11b-2H-hexahydro-4-pyrazino(2,1-a)isoquinolinones and intermediates ELF SANOFI (FR) 1983-08-24 EP disclosed