SCHEMBL11029433

SCHEMBL11029433

O=C1NCC(CCc2ccccc2)N(C(=O)C2CC2)C1=O

nearest known ligand 0.44

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SLC18A2 Q05940 1/20 0.43
KCNH2 Q12809 1/20 0.42
MTNR1B P49286 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11027618 0.84 KCNH2 (0.45) SLC18A2KCNH2
SCHEMBL11028695 0.79 KCNH2 (0.39) KCNH2
SCHEMBL11030839 0.72 SLC18A2 (0.40) SLC18A2KCNH2
SCHEMBL4664890 0.69 MTNR1B (0.40) MTNR1B
SCHEMBL11024548 0.68 MTNR1B (0.42) SLC18A2KCNH2MTNR1B
SCHEMBL11031319 0.65 SLC18A2 (0.42) SLC18A2
SCHEMBL11025726 0.65 TACR2 (0.44)
SCHEMBL11288045 0.64 ATM (0.51) SLC18A2
SCHEMBL28328103 0.64 ABCB1 (0.60) SLC18A2KCNH2MTNR1B
SCHEMBL14548187 0.63 FAAH (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0086678-B1 PROCESS FOR THE PREPARATION OF 2-ACYL-1,3,4,6,7,11B-2H-HEXAHYDRO-4-PYRAZINO(2,1-A)ISOQUINOLINONES AND INTERMEDIATES ELF SANOFI (FR) 1985-07-03 EP disclosed