SCHEMBL11033010

SCHEMBL11033010

CCCCCn1c(=O)c2[nH]c(O)nc2n(O)c1=O

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 2/20 0.48
ADORA1 P30542 3/20 0.46
SIRT1 Q96EB6 1/20 0.44
SIRT3 Q9NTG7 1/20 0.44
SIRT5 Q9NXA8 1/20 0.44
ADORA2A P29274 2/20 0.43
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31668890 0.77 ADORA2A (0.55) ADORA2BSIRT1SIRT3SIRT5ADORA2A
SCHEMBL11029795 0.75 ADORA2B (0.46) ADORA2BADORA1ADORA2APDE4APDE4B
SCHEMBL3120638 0.71 ADORA2B (0.49) ADORA2BADORA1SIRT1SIRT3SIRT5
SCHEMBL3114983 0.71 ADORA1 (0.53) ADORA2BADORA1SIRT1SIRT3SIRT5
SCHEMBL3119443 0.70 SIRT1 (0.54) ADORA2BADORA1SIRT1SIRT3SIRT5
SCHEMBL3117132 0.70 ADORA2B (0.51) ADORA2BADORA1SIRT1SIRT3SIRT5
SCHEMBL5405416 0.70 ADORA2A (0.54) ADORA2BADORA1SIRT1SIRT3SIRT5
SCHEMBL7918903 0.70 ADORA1 (0.57) ADORA2BADORA1SIRT1SIRT3SIRT5
SCHEMBL7022635 0.70 SIRT1 (0.56) ADORA2BADORA1SIRT1SIRT3SIRT5
SCHEMBL13247926 0.69 ADORA2B (0.53) ADORA2BADORA1SIRT1SIRT3SIRT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0075850-B1 PHARMACEUTICAL PREPARATIONS CONTAINING VICINAL DIHYDROXYALKYL XANTHINES, PROCESS FOR THE PREPARATION OF THE XANTHINES AND THE APPROPRIATE INTERMEDIATES THEREFOR HOECHST AKTIENGESELLSCHAFT (DE) 1985-12-18 EP claimed