SCHEMBL11033593

SCHEMBL11033593

CCOC(=O)n1c(=O)n(C2CCNCC2)c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
GAA P10253 2/20 0.48
L3MBTL1 Q9Y468 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2D6 P10635 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CHRM2 P08172 1/20 0.46
CHRM4 P08173 1/20 0.46
CHRM5 P08912 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.45
LMNA P02545 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11033286 0.82 HTR4 (0.45) MEN1KMT2AALDH1A1OPRM1
SCHEMBL11030825 0.82 CHRM2 (0.51) MEN1KMT2AGAAL3MBTL1CHRM2
SCHEMBL6577940 0.81 CHRM1 (0.67) MEN1KMT2AGAAL3MBTL1CHRM2
SCHEMBL4921218 0.78 OPRM1 (0.66) L3MBTL1ALDH1A1KDM4ETACR1OPRM1
SCHEMBL10268206 0.78 MEN1 (0.66) MEN1KMT2AGAAL3MBTL1CYP1A2
SCHEMBL2994414 0.78 HTR2C (0.42) CYP2C19CHRM2CHRM4CHRM5CHRM1
SCHEMBL13243414 0.77 OPRL1 (0.45) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL8060424 0.76 OPRL1 (0.60) OPRM1
SCHEMBL15642774 0.76 NOD2 (0.50) MEN1KMT2AL3MBTL1CHRM2CHRM4
SCHEMBL7582926 0.75 OPRL1 (0.52) CYP3A4TACR1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4446141-A Hypotensive piperidine derivatives KYOWA HAKKO KOGYO CO. (JP) 1984-05-01 US disclosed
EP-0018417-B1 NOVEL PIPERIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM KYOWA HAKKO KOGYO CO., LTD (JP) 1982-06-30 EP disclosed
EP-0018417-A1 Novel piperidine derivatives and pharmaceutical compositions containing them KYOWA HAKKO KOGYO CO., LTD (JP) 1980-11-12 EP disclosed