SCHEMBL11036058

SCHEMBL11036058

C=CCSc1nc(=O)n(CC2(C)CCCC2)c(=O)[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.40
HPGD P15428 6/20 0.40
PKM P14618 1/20 0.37
LMNA P02545 1/20 0.37
RAB9A P51151 1/20 0.37
RECQL P46063 1/20 0.36
HSD17B10 Q99714 3/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
POLB P06746 3/20 0.33
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TSHR P16473 1/20 0.32
GAA P10253 1/20 0.32
MAPK1 P28482 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11036035 0.74 ALDH1A1 (0.40) ALDH1A1HPGDPKMLMNARAB9A
SCHEMBL11040125 0.73 P2RX3 (0.30)
SCHEMBL14147928 0.64
SCHEMBL11020364 0.64 PDE4A (0.32) HPGDHSD17B10
SCHEMBL11021706 0.61 POLB (0.32) RAB9AMAPTMEN1KMT2APOLB
SCHEMBL11020046 0.61 P2RX3 (0.33) ALDH1A1
SCHEMBL9247800 0.60 ALDH1A1 (0.50) ALDH1A1HPGDPKMLMNARAB9A
SCHEMBL11846011 0.58 HCAR1 (0.39) ALDH1A1HPGD
SCHEMBL17767280 0.57 ALDH1A1 (0.47) ALDH1A1HPGDPKMRECQLHSD17B10
SCHEMBL11036030 0.57 P2RX3 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0160208-A1 3-(2,2-Tetramethylenepropyl)-1,3,5-triazine-2,4-diones BAYER AG (DE) 1985-11-06 EP claimed
EP-0160208-A1 3-(2,2-Tetramethylenepropyl)-1,3,5-triazine-2,4-diones BAYER AG (DE) 1985-11-06 EP disclosed