SCHEMBL11038869

SCHEMBL11038869

COc1cc2c(c(OC)c1OC)C=CN=C(N)C2

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.37
MAPT P10636 2/20 0.36
CYP3A4 P08684 1/20 0.36
POLB P06746 2/20 0.36
KDM4E B2RXH2 2/20 0.36
PDE5A O76074 1/20 0.35
ADORA1 P30542 1/20 0.35
TDP1 Q9NUW8 2/20 0.34
ACHE P22303 2/20 0.34
GAA P10253 1/20 0.34
LMNA P02545 1/20 0.34
ALOX5 P09917 1/20 0.33
TSHR P16473 1/20 0.33
APOBEC3A P31941 1/20 0.33
HTT P42858 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11038861 0.98 ATM (0.36) ATMMAPTCYP3A4POLBKDM4E
SCHEMBL11041640 0.76 BRD4 (0.45) MAPTCYP3A4KDM4EGAA
SCHEMBL11043192 0.76 ATM (0.37) ATMMAPTCYP3A4POLBKDM4E
SCHEMBL11039921 0.76 LMNA (0.43) ATMMAPTCYP3A4POLBKDM4E
Hydrochloric Acid SCHEMBL11040043 0.75 BRD4 (0.44) MAPTCYP3A4POLBKDM4EGAA
SCHEMBL11060113 0.74 ADORA1 (0.31) ADORA1ACHE
Hydrochloric Acid SCHEMBL11056785 0.69 ADRA1A (0.37) MAPTCYP3A4KDM4EACHEGAA
SCHEMBL11040367 0.69 MAPT (0.40) MAPTCYP3A4KDM4EGAALMNA
SCHEMBL11057303 0.69 MAPT (0.40) MAPTCYP3A4KDM4EGAALMNA
Hydrochloric Acid SCHEMBL11038881 0.69 BRD4 (0.38) MAPTCYP3A4POLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0115961-A2 Process for preparing benzazepines ELI LILLY AND COMPANY (US) 1984-08-15 EP claimed
EP-0116444-A2 Improvements in or relating to benzazepine derivatives ELI LILLY AND COMPANY (US) 1984-08-22 EP disclosed