SCHEMBL11040085

SCHEMBL11040085

NS(=O)(=O)c1cc(Nc2ccc3c(c2)C(C(=O)OCc2ccccc2)NCC3)ccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX4 Q99571 2/20 0.40
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA12 O43570 2/20 0.39
CA9 Q16790 2/20 0.39
ENPP2 Q13822 3/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KCNA5 P22460 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
GPR55 Q9Y2T6 1/20 0.36
CA3 P07451 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA13 Q8N1Q1 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11282932 0.89 NPC1 (0.53) CA1CA2CA12CA9NPC1
SCHEMBL11211694 0.84 ENPP2 (0.36) CA1CA2CA12CA9ENPP2
SCHEMBL11040082 0.81 P2RX4 (0.40) P2RX4CA1CA2CA12CA9
SCHEMBL11028997 0.76 TSHR (0.45) NPSR1
SCHEMBL11282929 0.71 NPC1 (0.53) CA1CA2CA12CA9NPC1
SCHEMBL19398221 0.69 TSHR (0.44) CA1CA2NPSR1
SCHEMBL11037355 0.68 ENPP2 (0.42) P2RX4CA1CA2CA12CA9
SCHEMBL15654433 0.67 ALDH1A1 (0.47) CA1CA2NPSR1
SCHEMBL4554597 0.67 TSHR (0.42) NPSR1
SCHEMBL19225930 0.65 TSHR (0.44) KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0088350-B1 CARBOXYALKYL DIPEPTIDES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SCHERING CORPORATION (US) 1985-02-20 EP disclosed