SCHEMBL11028997

SCHEMBL11028997

Nc1ccc2c(c1)C(C(=O)OCc1ccccc1)NCC2

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
MAPKAPK2 P49137 1/20 0.41
GLA P06280 1/20 0.41
FABP7 O15540 1/20 0.40
FABP5 Q01469 1/20 0.40
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC22A1 O15245 1/20 0.39
PRCP P42785 1/20 0.39
BACE1 P56817 1/20 0.39
ADRB2 P07550 1/20 0.38
KDM1A O60341 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11024334 0.83 KMT2A (0.40) TSHRNPSR1SLC6A2SLC6A4
SCHEMBL19398221 0.80 TSHR (0.44) TSHRNPSR1MAPKAPK2ADRB2KDM1A
SCHEMBL22080378 0.79 CYP3A4 (0.41) TSHRFABP7FABP5
SCHEMBL6967406 0.78 TSHR (0.42) TSHRNPSR1MAPKAPK2SLC6A2SLC6A4
SCHEMBL4554597 0.78 TSHR (0.42) TSHRNPSR1MAPKAPK2GLAADRB2
SCHEMBL7202686 0.78 TSHR (0.62) TSHRNPSR1MAPKAPK2SLC6A2SLC6A4
SCHEMBL19225930 0.76 TSHR (0.44) TSHRNPSR1MAPKAPK2GLAFABP7
SCHEMBL7436594 0.76 GLA (0.44) TSHRMAPKAPK2GLAFABP7FABP5
SCHEMBL11040085 0.76 P2RX4 (0.40) NPSR1
SCHEMBL15654433 0.74 ALDH1A1 (0.47) TSHRNPSR1SLC6A2SLC6A4SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0088350-B1 CARBOXYALKYL DIPEPTIDES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SCHERING CORPORATION (US) 1985-02-20 EP disclosed
EP-0088350-A1 Carboxyalkyl dipeptides, processes for their production and pharmaceutical compositions containing them SCHERING CORPORATION (US) 1983-09-14 EP disclosed