SCHEMBL11041232

SCHEMBL11041232

COC(=O)Oc1nnn(-c2ccc([N+](=O)[O-])cc2)c1N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.49
TP53 P04637 1/20 0.48
MAPT P10636 6/20 0.47
ALDH1A1 P00352 5/20 0.47
KDM4E B2RXH2 2/20 0.46
IDO1 P14902 1/20 0.44
TDO2 P48775 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
NPC1 O15118 1/20 0.44
NFKB1 P19838 1/20 0.44
RAB9A P51151 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
SLC5A1 P13866 1/20 0.43
SLC5A2 P31639 1/20 0.43
MEN1 O00255 1/20 0.42
PKM P14618 1/20 0.41
LMNA P02545 2/20 0.41
HPGD P15428 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11038855 0.83 TP53 (0.63) KMT2ATP53ALDH1A1SMN1; SMN2NPC1
SCHEMBL11096860 0.82 SMN1; SMN2 (0.55) TP53ALDH1A1KDM4ESMN1; SMN2LMNA
SCHEMBL11044738 0.82 TP53 (0.49) TP53ALDH1A1IDO1TDO2SMN1; SMN2
SCHEMBL11095871 0.81 TP53 (0.54) KMT2ATP53ALDH1A1KDM4EIDO1
SCHEMBL10985550 0.81 TP53 (0.69) KMT2ATP53MAPTALDH1A1KDM4E
SCHEMBL11040213 0.77 IDO1 (0.43) KMT2ATP53MAPTALDH1A1IDO1
SCHEMBL11044671 0.76 POLB (0.49) KMT2ATP53MAPTALDH1A1SMN1; SMN2
SCHEMBL11047507 0.75 MAPT (0.43) KMT2ATP53MAPTALDH1A1SMN1; SMN2
SCHEMBL11042738 0.69 SMN1; SMN2 (0.49) KMT2ATP53MAPTALDH1A1KDM4E
SCHEMBL84030 0.69 GAA (0.62) KMT2ATP53MAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0073931-B1 ANILINO-1,2,3-TRIAZOLE DERIVATIVES, MEDICAMENTS CONTAINING THEM, PROCESS FOR PREPARING THEM, AND THEIR USE BOEHRINGER INGELHEIM KG (DE) 1985-02-13 EP disclosed
EP-0073931-A1 Anilino-1,2,3-triazole derivatives, medicaments containing them, process for preparing them, and their use BOEHRINGER INGELHEIM KG (DE) 1983-03-16 EP disclosed