SCHEMBL11042341

SCHEMBL11042341

C=C(C)c1cc(F)ccc1F

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.56
CES1 P23141 3/20 0.56
CA3 P07451 1/20 0.44
CA6 P23280 1/20 0.44
CA5A P35218 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
CA5B Q9Y2D0 1/20 0.44
HRH4 Q9H3N8 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
TAS1R2 Q8TE23 1/20 0.36
KEAP1 Q14145 1/20 0.36
ALDH1A1 P00352 5/20 0.35
MDM2 Q00987 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21207989 0.84 CES2 (0.41) CES2CES1CA3CA6CA5A
SCHEMBL29727310 0.82 CES2 (0.56) CES2CES1CA3CA6CA5A
SCHEMBL13689710 0.82 CES2 (0.56) CES2CES1CA3CA6CA5A
SCHEMBL16960709 0.81 CES2 (0.60) CES2CES1CA3CA6CA5A
SCHEMBL19859386 0.80 CLK1 (0.40) CES2CES1CA3CA6CA5A
SCHEMBL15177920 0.80 NFE2L2 (0.39) CES2CES1ALDH1A1TSHRMAPK1
SCHEMBL10290613 0.80 CA3 (0.43) CES2CES1CA3CA6CA5A
SCHEMBL15172864 0.80 CES2 (0.39) CES2CES1CA3CA6CA5A
SCHEMBL16959306 0.79 CES2 (0.58) CES2CES1CA3CA6CA5A
SCHEMBL23864570 0.78 ALDH1A1 (0.35) CES2CES1HRH4ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0030716-B1 CHLORINATED PVC BLENDS WITH IMPROVED PROCESSABILITY The B.F. GOODRICH Company (US) 1984-02-08 EP claimed
US-8916593-B2 Alkoxy-substituted 2-aminopyridines as ALK inhibitors PFIZER INC. (US) 2014-12-23 US disclosed
US-20130196952-A1 HETEROCYCLIC DERIVATIVES FOR THE TREATMENT OF DISEASES PFIZER INC. (US) 2013-08-01 US disclosed
WO-2009061596-A1 COMPOUNDS FOR INHIBITING KSP KINESIN ACTIVITY SCHERING CORPORATION (US) 2009-05-14 WO disclosed
WO-2009052288-A1 SPIRO-CONDENSED 1, 3, 4-THIADIAZOLE DERIVATIVES FOR INHIBITING KSP KINESIN ACTIVITY SCHERING CORPORATION (US) 2009-04-23 WO disclosed
EP-1697336-B1 AROYLFURANES AND AROYLTHIOPHENES SUITABLE FOR THE TREATMENT OF CANCER BASILEA PHARMACEUTICA AG (CH) 2007-12-19 EP disclosed
WO-2007062308-A2 HOMO- AND HETEROCYCLIC COMPOUNDS SUITABLE AS CETP INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-31 WO disclosed
EP-0030716-B1 CHLORINATED PVC BLENDS WITH IMPROVED PROCESSABILITY The B.F. GOODRICH Company (US) 1984-02-08 EP disclosed
US-4304884-A A-ALKYLSTYRENE-VINYLBENZENE OR ACRYLATE-NITRILE TERPOLYMER THE B. F. GOODRICH COMPANY (US) 1981-12-08 US disclosed
EP-0030716-A1 Chlorinated PVC blends with improved processability The B.F. GOODRICH Company (US) 1981-06-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130196952-A1 HETEROCYCLIC DERIVATIVES FOR THE TREATMENT OF DISEASES ALK, ETV6, ACVR1 CES2 2687/4885CES1 1172/4885CA3 4701/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.